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Digoxin pharmacokinetics and MDR1 genetic polymorphisms

Author
VERSTUYFT, Céline1 ; SCHWAB, Mathias2 ; SCHAEFFELER, Elke2 ; KERB, Reinhold3 ; BRINKMANN, Ulrich3 ; JAILLON, Patrice1 4 ; FUNCK-BRENTANO, Christian1 4 ; BECQUEMONT, Laurent1
[1] Department of Pharmacology, Saint-Antoine Hospital, 184 rue du Faubourg Saint Antoine, 75012, Paris, France
[2] Dr. Margarete Fischer-Bosch-Institut für Klinische Pharmakologie, Auerbachstrasse 112, 70376, Stuttgart, Germany
[3] Epidauros Biotechnologie AG, Am Neuland 1, 82347, Bernried, Germany
[4] Clinical Investigation Center, Saint-Antoine Hospital, 184 rue du Faubourg Saint Antoine, Paris, France
Source

European journal of clinical pharmacology. 2003, Vol 58, Num 12, pp 809-812, 4 p ; ref : 14 ref

ISSN
0031-6970
Scientific domain
Pharmacology drugs
Publisher
Springer, Berlin / Springer, Heidelberg
Publication country
Germany
Document type
Article
Language
English
Author keyword
Digoxin Genetic polymorphism Human MDR1 P-glycoprotein
Keyword (fr)
Cardiotonique Caucasoïde Digitalique Digoxine Expression génique Français Glycoprotéine P Glycoside Homme Individu sain Métabolisme Pharmacocinétique Pharmacogénétique Phénotype Polymorphisme mononucléotide Voie orale Gène MDR1 Génétique
Keyword (en)
Cardiotonic agent Caucasoid Digitalis drug Digoxin Gene expression French P Glycoprotein Glycoside Human Healthy subject Metabolism Pharmacokinetics Pharmacogenetics Phenotype Single nucleotide polymorphism Oral administration Genetics
Keyword (es)
Cardiotónico Caucásico Digitálico Digoxina Expresión genética Francés Glicoproteína P Glicósido Hombre Individuo sano Metabolismo Farmacocinética Farmacogenética Fenotipo Polimorfismo mononucleótido Vía oral Genética
Classification
Pascal
002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02F Cardiovascular system / 002B02F01 Cardiotonic agents

Discipline
Pharmacological treatments
Origin
Inist-CNRS
Database
PASCAL
INIST identifier
14728164

Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS

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