Potent small molecule CCR1 antagonists
- Author
- KATH, John C1 ; BRISSETTE, William H1 ; MARTIN, William H1 ; MCELROY, Eric B1 ; MCGLYNN, Molly A1 ; PARADIS, Timothy J1 ; POSS, Christopher S1 ; STOCK, Ingrid A1 ; TYLASKA, Laurie A1 ; DEYE ZHENG1 ; BROWN, Matthew F1 ; CONKLYN, Maryrose1 ; DIRICO, Amy P1 ; DORFF, Peter1 ; GLADUE, Ronald P1 ; LILLIE, Brett M1 ; LIRA, Paul D1 ; MAIRS, Erin N1
[1] Pfizer Global Research and Development, Eastern Point Road, Groton, CT 06340, United States - Source
Bioorganic & medicinal chemistry letters (Print). 2004, Vol 14, Num 9, pp 2169-2173, 5 p
- ISSN
- 0960-894X
- Scientific domain
- Biochemistry, molecular biology, biophysics; Pharmacology drugs
- Publisher
- Elsevier, Oxford
- Publication country
- United Kingdom
- Document type
- Article
- Language
- English
- Keyword (fr)
- Alcool Antagoniste Carboxamide Composé peptidomimétique In vitro Quinoxaline dérivé Relation structure activité Récepteur chimiokine CCR1 Synthèse chimique Hexanamide(4-hydroxy-2-isopentyl-6-phényl-5-[quinoxalin-2-ylcarbonylamino])
- Keyword (en)
- Alcohol Antagonist Carboxamide Peptidomimetic compound In vitro Quinoxaline derivatives Structure activity relation CCR1 chemokine receptor Chemical synthesis
- Keyword (es)
- Alcohol Antagonista Carboxamida Compuesto peptidomimético In vitro Quinoxalina derivado Relación estructura actividad Receptor quimioquina CCR1 Síntesis química
- Classification
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02Q Immunomodulators
- Discipline
- Pharmacological treatments
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 15695760
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1016/j.bmcl.2004.02.021 
https://dx.doi.org/10.1016/j.bmcl.2004.02.021
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