Novel retinoid X receptor (RXR) antagonists having a dicarba-closo-dodecaborane as a hydrophobic moiety
- Author
- OHTA, Kiminori1 ; IIJIMA, Toru2 ; KAWACHI, Emiko2 ; KAGECHIKA, Hiroyuki2 ; ENDO, Yasuyuki1
[1] Faculty of Pharmaceutical Sciences, Tohoku Pharmaceutical University, 4-4-1, Komatsushima, Aoba-ku, Sendai 981-8558, Japan
[2] Graduate School of Pharmaceutical Sciences, The University of Tokyo, 7-3-1, Hongo, Bunkyo-ku, Tokyo 113-0033, Japan - Source
Bioorganic & medicinal chemistry letters (Print). 2004, Vol 14, Num 23, pp 5913-5918, 6 p
- ISSN
- 0960-894X
- Scientific domain
- Biochemistry, molecular biology, biophysics; Pharmacology drugs
- Publisher
- Elsevier, Oxford
- Publication country
- United Kingdom
- Document type
- Article
- Language
- English
- Keyword (fr)
- Activité biologique Antagoniste Bore composé organique Carborane Cellule tumorale Composé cage Cytodifférenciation Homme Hétérodimère Leucémie Lignée HL60 Lignée cellulaire Récepteur acide rétinoïque RAR Récepteur rétinoïde RXR Synthèse chimique Sélectivité Dicarba-closo-dodécaborane dérivé Hémopathie maligne
- Keyword (en)
- Biological activity Antagonist Organic boron compounds Carborane Tumor cell Cage compound Cell differentiation Human Heterodimer Leukemia HL60 cell line Cell line RAR retinoic acid receptor RXR retinoid receptor Chemical synthesis Selectivity Malignant hemopathy
- Keyword (es)
- Actividad biológica Antagonista Carborano Célula tumoral Compuesto jaula Diferenciación celular Hombre Heterodimero Leucemia Línea HL60 Línea celular Receptor ácido retinoico RAR Receptor retinoide RXR Síntesis química Selectividad Hemopatía maligna
- Classification
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02B Neuropharmacology / 002B02B09 Neurotransmitters. Neurotransmission. Receptors / 002B02B09G Miscellaneous
- Discipline
- Pharmacological treatments
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 16223744
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1016/j.bmcl.2004.09.035 
https://dx.doi.org/10.1016/j.bmcl.2004.09.035
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