Synthesis and in vitro selective anti-Helicobacter pylori activity of pyrazoline derivatives
- Author
- CHIMENTI, F1 ; BIZZARRI, B1 ; BRENCIAGLIA, M. I2 ; MANNA, F1 ; BOLASCO, A1 ; SECCI, D1 ; CHIMENTI, P1 ; GRANESE, A1 ; RIVANERA, D2 ; LILLI, D2 ; SCALTRITO, M. M3
[1] Dipartimento di Studi di Chimica e Tecnologia delle Sostanze Biologicamente Attive, Univesità ' La Sapienza', P. le A. Moro 5, 00185 Rome, Italy
[2] Dipartimento di Scienze di Sanità Pubblica, Università ' La Sapienza', P.le A. Moro 5, 00185 Rome, Italy
[3] Istituto di Microbiologia, Università degli Studi di Milano, via Pascal 36, 20133 Milano, Italy - Source
Bioorganic & medicinal chemistry letters (Print). 2005, Vol 15, Num 3, pp 603-607, 5 p
- ISSN
- 0960-894X
- Scientific domain
- Biochemistry, molecular biology, biophysics; Pharmacology drugs
- Publisher
- Elsevier, Oxford
- Publication country
- United Kingdom
- Document type
- Article
- Language
- English
- Keyword (fr)
- Activité biologique Antibactérien Helicobacter pylori In vitro Métronidazole Phénols Pyrazole dérivé Résistance Synthèse chimique Sélectivité Pyrazole(1-acétyl-4,5-dihydro-3-[4-hydroxyphényl]-5-[p-tolyl]) Bactérie Spirillaceae Spirillales
- Keyword (en)
- Biological activity Antibacterial agent Helicobacter pylori In vitro Metronidazole Phenols Pyrazole derivatives Resistance Chemical synthesis Selectivity Bacteria Spirillaceae Spirillales
- Keyword (es)
- Actividad biológica Antibacteriano Helicobacter pylori In vitro Metronidazol Fenoles Pirazol derivado Resistencia Síntesis química Selectividad Bacteria Spirillaceae Spirillales
- Classification
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02S Antibiotics. Antiinfectious agents. Antiparasitic agents / 002B02S02 Antibacterial agents
- Discipline
- Pharmacological treatments
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 16478186
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1016/j.bmcl.2004.11.042 
https://dx.doi.org/10.1016/j.bmcl.2004.11.042
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