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TARP auxiliary subunits switch AMPA receptor antagonists into partial agonists

Author
MENUZ, Karen1 2 ; STROUD, Robert M3 ; NICOLL, Roger A1 4 ; HAYS, Franklin A3
[1] Department of Cellular and Molecular Pharmacology, University of California at San Francisco, San Francisco, CA 94143, United States
[2] Graduate Program in Neuroscience, University of California at San Francisco, San Francisco, CA 94143, United States
[3] Department of Biochemistry and Biophysics, University of California at San Francisco, San Francisco, CA 94143, United States
[4] Department of Physiology, University of California at San Francisco, San Francisco, CA 94143, United States
Source

Science (Washington, D.C.). 2007, Vol 318, Num 5851, pp 815-817, 3 p ; ref : 33 ref

CODEN
SCIEAS
ISSN
0036-8075
Scientific domain
Multidisciplinary
Publisher
American Association for the Advancement of Science, Washington, DC
Publication country
United States
Document type
Article
Language
English
Keyword (fr)
Agoniste partiel Antagoniste Fixation ligand Neurone Protéine transmembranaire Récepteur AMPA Sousunité Système nerveux central Récepteur glutamate
Keyword (en)
Partial agonist Antagonist Ligand binding Neuron Transmembrane protein AMPA receptor Subunit Central nervous system Glutamate receptor
Keyword (es)
Agonista parcial Antagonista Fijación ligando Neurona Proteína transmembranar Receptor AMPA Subunitad Sistema nervioso central Receptor glutámato
Classification
Pascal
002 Biological and medical sciences / 002A Fundamental and applied biological sciences. Psychology / 002A04 Molecular and cellular biology / 002A04F Cell structures and functions / 002A04F03 Cell receptors / 002A04F03C Aminoacid receptors (glycine, glutamate, gaba)

Discipline
Molecular and cell biology
Origin
Inist-CNRS
Database
PASCAL
INIST identifier
19219187

Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS

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