Synthesis and biological evaluation of N-antipyrine-4-substituted amino-3-chloromaleimide derivatives
- Author
- MAHLE, Fernanda1 ; GUIMARAES, Tatiana da Rosa1 ; VERGILINA MEIRA, Aleandra1 ; CORREA, Rogério1 ; CE BELLA CRUZ, Rosana1 ; CRUZ, Alexandre Bella1 ; NUNES, Ricardo José2 ; CECHINEL-FILHO, Valdir1 ; DE CAMPOS-BUZZI, Fátima1
[1] Núcleo de Investigações Químico-Farmacêuticas (NIQFAR)/CCS, Universidade do Vale do Itajaf (UNIVALI), Caixa Postal 360, CEP 88302-202, Itajaí, Santa Catarina, Brazil
[2] Departamento de Quimica, Curso de Pós-Graduação em Química, Universidade Federal de Santa Catarina, UFSC, Florianópolis, Brazil - Source
European journal of medicinal chemistry. 2010, Vol 45, Num 11, pp 4761-4768, 8 p ; ref : 27 ref
- CODEN
- EJMCA5
- ISSN
- 0223-5234
- Scientific domain
- Organic chemistry; Pharmacology drugs
- Publisher
- Elsevier, Kidlington
- Publication country
- United Kingdom
- Document type
- Article
- Language
- English
- Author keyword
- Antimicrobial activity Antinociceptive activity Antipyrine Cyclic imides
- Keyword (fr)
- Amine aromatique Amine Analgésique Animal Antibactérien Antifongique Antimicrobien Cycle 5 chaînons Dérivé de l'aniline Hétérocycle azote Imide In vitro In vivo Relation structure activité Souris Synthèse chimique Antipyrine dérivé Maléimide dérivé Pyrazol-3-one dérivé Mammalia Rodentia Vertebrata
- Keyword (en)
- Aromatic amine Amine Analgesic Animal Antibacterial agent Antifungal agent Antimicrobial agent Five membered ring Aniline derivatives Nitrogen heterocycle Imide In vitro In vivo Structure activity relation Mouse Chemical synthesis Mammalia Rodentia Vertebrata
- Keyword (es)
- Amina aromática Amina Analgésico Animal Antibacteriano Antifúngico Antimicrobiano Ciclo 5 eslabones Anilina derivado Heterociclo nitrógeno Imida In vitro In vivo Relación estructura actividad Ratón Síntesis química Mammalia Rodentia Vertebrata
- Classification
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02B Neuropharmacology / 002B02B05 Analgesics
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02S Antibiotics. Antiinfectious agents. Antiparasitic agents / 002B02S01 General aspects
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02S Antibiotics. Antiinfectious agents. Antiparasitic agents / 002B02S02 Antibacterial agents
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02S Antibiotics. Antiinfectious agents. Antiparasitic agents / 002B02S04 Antifungal agents
- Discipline
- Pharmacological treatments
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 23367489
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1016/j.ejmech.2010.07.040 
https://dx.doi.org/10.1016/j.ejmech.2010.07.040
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