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An investigation of the safety and pharmacokinetics of the novel TRPV1 antagonist XEN-D0501 in healthy subjects

Author
ROUND, Patrick1 ; PRIESTLEY, Anthony2 ; ROBINSON, Jan1
[1] Xention Ltd, United Kingdom
[2] LCG Bioscience, Combridge, United Kingdom
Source

British journal of clinical pharmacology. 2011, Vol 72, Num 6, pp 921-931, 11 p ; ref : 29 ref

CODEN
BCPHBM
ISSN
0306-5251
Scientific domain
Pharmacology drugs
Publisher
Blackwell, Oxford
Publication country
United Kingdom
Document type
Article
Language
English
Author keyword
TRPV1 antagonist XEN-D0501 overactive bladder
Keyword (fr)
Antagoniste Homme Individu sain Pharmacocinétique Récepteur vanilloïde VR1 Sécurité Toxicité Vessie hyperactive Récepteur vanilloïde TRPV1 Pathologie de l'appareil urinaire Pathologie de la vessie Pathologie des voies urinaires
Keyword (en)
Antagonist Human Healthy subject Pharmacokinetics VR1 vanilloid receptor Safety Toxicity Overactive bladder TRPV1 vanilloid receptor Urinary system disease Bladder disease Urinary tract disease
Keyword (es)
Antagonista Hombre Individuo sano Farmacocinética Receptor vaniloide VR1 Seguridad Toxicidad Vejiga hiperactiva Aparato urinario patología Vejiga patología Vía urinaria patología
Classification
Pascal
002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments

Pascal
002 Biological and medical sciences / 002B Medical sciences / 002B14 Nephrology. Urinary tract diseases / 002B14E Urinary system involvement in other diseases. Miscellaneous / 002B14E02 Urinary tract. Prostate gland

Discipline
General pharmacology Nephrology. Urinary tract diseases
Origin
Inist-CNRS
Database
PASCAL
INIST identifier
24756278

Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS

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