Family-wide chemical profiling and structural analysis of PARP and tankyrase inhibitors
- Author
- WAHLBERG, Elisabet1 ; KARLBERG, Tobias1 ; KULL, Björn4 ; ROBERTSON, Graeme Michael2 ; PELLICCIARI, Roberto2 ; SCHÜLER, Herwig1 ; WEIGELT, Johan1 ; KOUZNETSOVA, Ekaterina1 ; MARKOVA, Natalia1 ; MACCHIARULO, Antonio2 ; THORSELL, Ann-Gerd1 ; POL, Ewa3 ; FROSTELL, Asa3 ; EKBLAD, Torun1 ; ÖNCÜ, Delal4
[1] Structural Genomics Consortium, Karolinska Institutet, Department of Medical Biochemistry and Biophysics, Stockholm, Sweden
[2] Dipartimento di Chimica e Tecnologia del Farmaco, University of Perugia, Perugia, Italy
[3] GE Healthcare Bio-Sciences AB, Uppsala, Sweden
[4] Actar AB, Stockholm, Sweden - Source
Nature biotechnology (Print). 2012, Vol 30, Num 3, pp 283-288, 6 p ; ref : 43 ref
- CODEN
- NABIF9
- ISSN
- 1087-0156
- Scientific domain
- Biotechnology
- Publisher
- Nature Publishing Group, New York, NY
- Publication country
- United States
- Document type
- Article
- Language
- English
- Keyword (fr)
- Analyse structurale Anticancéreux Inhibiteur enzyme NAD+ ADP-ribosyltransferase Spécificité Tankyrase Enzyme Glycosyltransferases Pentosyltransferases Transferases
- Keyword (en)
- Structural analysis Antineoplastic agent Enzyme inhibitor NAD+ ADP-ribosyltransferase Specificity Enzyme Glycosyltransferases Pentosyltransferases Transferases
- Keyword (es)
- Análisis estructural Anticanceroso Inhibidor enzima NAD+ ADP-ribosyltransferase Especificidad Enzima Glycosyltransferases Pentosyltransferases Transferases
- Classification
- Pascal
- 002 Biological and medical sciences / 002A Fundamental and applied biological sciences. Psychology / 002A31 Biotechnology
- Discipline
- Biotechnology
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 25626588
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1038/nbt.2121 
https://dx.doi.org/10.1038/nbt.2121
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