Synthesis and evaluation of analogues of estrone-3-O-sulfamate as potent steroid sulfatase inhibitors
- Author
- LAWRENCE WOO, L. W1 ; LEBLOND, Bertrand1 ; PUROHIT, Atul2 ; POTTER, Barry V. L1
[1] Medicinal Chemistry, Department of Pharmacy & Pharmacology, University of Bath, Claverton Down, Bath BA2 7AY, United Kingdom
[2] Diabetes, Endocrinology & Metabolism, Imperial College London, Section of Investigative Medicine, 6th Floor, Commonwealth Building (6N2B), Hammersmith Hospital, Du Cane Road, London W12 0NN, United Kingdom - Source
Bioorganic & medicinal chemistry. 2012, Vol 20, Num 8, pp 2506-2519, 14 p ; ref : 50 ref
- ISSN
- 0968-0896
- Scientific domain
- Biochemistry, molecular biology, biophysics; Pharmacology drugs
- Publisher
- Elsevier, Amsterdam
- Publication country
- Netherlands
- Document type
- Article
- Language
- English
- Author keyword
- Breast cancer EMATE Endocrine therapy Inhibitors Steroid sulfatase
- Keyword (fr)
- Amidosulfate organique Cancer du sein Estrone Evaluation Glande mammaire Inhibiteur enzyme Pathologie de la glande mammaire Steryl-sulfatase Synthèse chimique Traitement hormonal Tumeur maligne Inhibiteur steroid sulfatase Cancer Enzyme Esterases Hydrolases Pathologie du sein Sulfuric ester hydrolases
- Keyword (en)
- Organic amidosulfate Breast cancer Estrone Evaluation Mammary gland Enzyme inhibitor Mammary gland diseases Steryl-sulfatase Chemical synthesis Hormone therapy Malignant tumor Cancer Enzyme Esterases Hydrolases Breast disease Sulfuric ester hydrolases
- Keyword (es)
- Amidosulfato orgánico Cáncer del pecho Estrona Evaluación Glándula mamaria Inhibidor enzima Glándula mamaria patología Steryl-sulfatase Síntesis química Hormonoterapia Tumor maligno Cáncer Enzima Esterases Hydrolases Seno patología Sulfuric ester hydrolases
- Classification
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02A General pharmacology / 002B02A07 Miscellaneous
- Discipline
- General pharmacology
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 25855758
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1016/j.bmc.2012.03.007 
https://dx.doi.org/10.1016/j.bmc.2012.03.007
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