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New Chemical Scaffolds for Human African Trypanosomiasis Lead Discovery from a Screen of Tyrosine Kinase Inhibitor Drugs

Author
BEHERA, Ranjan1 ; THOMAS, Sarah M1 ; MENSA-WILMOT, Kojo1
[1] Department of Cellular Biology, University of Georgia, Athens, Georgia, United States
Source

Antimicrobial agents and chemotherapy. 2014, Vol 58, Num 4, pp 2202-2210, 9 p ; ref : 64 ref

CODEN
AACHAX
ISSN
0066-4804
Scientific domain
Microbiology, infectious diseases; Pharmacology drugs
Publisher
American Society for Microbiology, Washington, DC
Publication country
United States
Document type
Article
Language
English
Keyword (fr)
Antiparasitaire Homme Inhibiteur de la tyrosine kinase Inhibiteur enzyme Mécanisme action Protein-tyrosine kinase Trypanosoma brucei Trypanosomiase africaine Voie orale Enzyme Infection Kinetoplastida Parasitose Protozoa Protozoose Transferases Trypanosomiase
Keyword (en)
Parasiticide Human Tyrosine kinase inhibitor Enzyme inhibitor Mechanism of action Protein-tyrosine kinase Trypanosoma brucei African sickness Oral administration Enzyme Infection Kinetoplastida Parasitosis Protozoa Protozoal disease Transferases Trypanosomiasis
Keyword (es)
Antiparasitario Hombre Inhibidor tyrosine kinase Inhibidor enzima Mecanismo acción Protein-tyrosine kinase Trypanosoma brucei Tripanosomiasis africana Vía oral Enzima Infección Kinetoplastida Parasitosis Protozoa Protozoosis Transferases Tripanosomiasis
Classification
Pascal
002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02S Antibiotics. Antiinfectious agents. Antiparasitic agents / 002B02S06 Antiparasitic agents

Pascal
002 Biological and medical sciences / 002B Medical sciences / 002B05 Infectious diseases / 002B05E Parasitic diseases / 002B05E02 Protozoal diseases / 002B05E02B Human protozoal diseases / 002B05E02B6 Trypanosomiasis

Discipline
Infectious pathology Pharmacological treatments
Origin
Inist-CNRS
Database
PASCAL
INIST identifier
28416823

Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS

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