Antitrypanosomal Activity of Fexinidazole Metabolites, Potential New Drug Candidates for Chagas Disease
- Author
- BAHIA, Maria T1 ; NASCIMENTO, Alvaro F. S1 ; KOLTUN, Maria3 ; SAUNDERS, Jessica3 ; WHITE, Karen L3 ; SCANDALE, Ivan2 ; CHARMAN, Susan A3 ; CHATELAIN, Eric2 ; MAZZETI, Ana Lia1 ; MARQUES, Luiz F1 ; GONCALVES, Karolina R1 ; MOTA, Ludmilla W. R1 ; DINIZ, Lívia de F1 ; CALDAS, Ivo S1 ; TALVANI, André1 ; SHACKLEFORD, David M3
[1] Laboratório de Doença de Chagas, Departamento de Ciências Biológicas & Núcleo de Pesquisas em Ciências Biológicas, Universidade Federal de Ouro Preto, Campus Universitário Morro do Cruzeiro, Ouro Preto, Brazil
[2] Drugs for Neglected Diseases initiative, Geneva, Switzerland
[3] Centre for Drug Candidate Optimisation, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia - Source
Antimicrobial agents and chemotherapy. 2014, Vol 58, Num 8, pp 4362-4370, 9 p ; ref : 17 ref
- CODEN
- AACHAX
- ISSN
- 0066-4804
- Scientific domain
- Microbiology, infectious diseases; Pharmacology drugs
- Publisher
- American Society for Microbiology, Washington, DC
- Publication country
- United States
- Document type
- Article
- Language
- English
- Keyword (fr)
- Activité biologique Antiparasitaire Fexinidazole Métabolite Trypanosomiase américaine Nouveau médicament Infection Parasitose Protozoose Trypanosomiase
- Keyword (en)
- Biological activity Parasiticide Fexinidazole Metabolite Chagas disease Infection Parasitosis Protozoal disease Trypanosomiasis
- Keyword (es)
- Actividad biológica Antiparasitario Fexinidazol Metabolito Tripanosomiasis americana Infección Parasitosis Protozoosis Tripanosomiasis
- Classification
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02S Antibiotics. Antiinfectious agents. Antiparasitic agents
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B05 Infectious diseases / 002B05E Parasitic diseases / 002B05E02 Protozoal diseases / 002B05E02B Human protozoal diseases / 002B05E02B6 Trypanosomiasis
- Discipline
- Infectious pathology Pharmacological treatments
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 28691844
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1128/AAC.02754-13 
https://dx.doi.org/10.1128/AAC.02754-13
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