2-[(2-pyridylmethyl)sulfinyl]-1H-thieno[3,4-d]imidazoles. A novel class of gastric H+/K+-ATPase inhibitors
- Author
- WEIDMANN, K; HERLING, A. W; LANG, H.-J; SCHEUNEMANN, K.-H; RIPPEL, R; NIMMESGERN, H; SCHOLL, T; BICKEL, M; METZGER, H
Hoechst AG, pharma res., Frankfurt 6230, Germany - Source
Journal of medicinal chemistry (Print). 1992, Vol 35, Num 3, pp 438-450 ; ref : 51 ref
- CODEN
- JMCMAR
- ISSN
- 0022-2623
- Scientific domain
- Pharmacology drugs
- Publisher
- American Chemical Society, Washington, DC
- Publication country
- United States
- Document type
- Article
- Language
- English
- Keyword (fr)
- Composé bicyclique H+/K+-transporting ATPase Hétérocycle soufre azote In vitro In vivo Inhibiteur enzyme Relation structure activité Sulfoxyde Thiéno [2,3-d] imidazole(2-[2-pyridyl) méthane sulfinyl] Thiéno [3,4-d] imidazole(2-[(2-pyridyl) méthanesulfinyl]) Enzyme
- Keyword (en)
- Bicyclic compound H+/K+-transporting ATPase Sulfur nitrogen heterocycle In vitro In vivo Enzyme inhibitor Structure activity relation Sulfoxide Enzyme
- Keyword (es)
- Compuesto bicíclico H+/K+-transporting ATPase Heterociclo azufre nitrógeno In vitro In vivo Inhibidor enzima Relación estructura actividad Sulfóxido Enzima
- Classification
- Pascal
- 001 Exact sciences and technology / 001C Chemistry / 001C03 Organic chemistry / 001C03C Preparations and properties / 001C03C06 Heterocyclic compounds / 001C03C06D Heterocyclic compounds with n hetero atom and also o and/or s, se, te hetero atoms
- Discipline
- Organic chemistry
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 5189212
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1021/jm00081a004 
https://dx.doi.org/10.1021/jm00081a004
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