13,28-Epoxy triterpenoid saponins from Ardisia japonica selectively inhibit proliferation of liver cancer cells without affecting normal liver cellsQIN LI; WEI LI; HUI, Lin-Ping et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 19, pp 6120-6125, issn 0960-894X, 6 p.Article

2-(4-Chlorophenyl)-2-oxoethyl 4-benzamidobenzoate derivatives, a novel class of SENP1 inhibitors: Virtual screening, synthesis and biological evaluationYINGYI CHEN; DONGHUA WEN; ZHIMIN HUANG et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 22, pp 6867-6870, issn 0960-894X, 4 p.Article

3-Phenyl-1H-5-pyrazolylamine-based derivatives as potent and efficacious inhibitors of FMS-like tyrosine kinase-3 (FLT3)HSU, John T.-A; YEH, Teng-Kuang; CHANG, Yun-I et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 14, pp 4654-4659, issn 0960-894X, 6 p.Article

4-Arylphthalazin-1(2H)-one derivatives as potent antagonists of the melanin concentrating hormone receptor 1 (MCH-R1)CHAE JO LIM; SOO HEE KIM; BYUNG HO LEE et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 1, pp 427-430, issn 0960-894X, 4 p.Article

4-Phenoxypiperidine pyridazin-3-one histamine H₃ receptor inverse agonists demonstrating potent and robust wake promoting activityHUDKINS, Robert L; ZULLI, Allison L; RADDATZ, Rita et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 4, pp 1504-1509, issn 0960-894X, 6 p.Article

5-Benzothiazole substituted pyrimidine derivatives as HCV replication (replicase) inhibitorsARASAPPAN, Ashok; BENNETT, Frank; PINTO, Patrick et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 9, pp 3229-3234, issn 0960-894X, 6 p.Article

5-HT2c receptor selectivity and structure-activity relationship of N-methyl-N-(1-methylpiperidin-4-yl)benzenesulfonamide analogsJAE WAN JANG; BAEK, Je-Sook; GIL DON CHOI et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 1, pp 347-352, issn 0960-894X, 6 p.Article

6-Amino quinazolinedione sulfonamides as orally active competitive AMPA receptor antagonistsORAIN, David; OFNER, Silvio; FLOERSHEIM, Philipp et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 2, pp 996-999, issn 0960-894X, 4 p.Article

A DNA aptamer sensor for 8-oxo-7,8-dihydroguanineROY, Jyoti; CHIRANIA, Payal; GANGULY, Sanniv et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 2, pp 863-867, issn 0960-894X, 5 p.Article

A new antifungal and cytotoxic C-methylated flavone glycoside from Picea neoveitchiiCHEN, Wei-Quan; SONG, Zhi-Jun; XU, Han-Hong et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 18, pp 5819-5822, issn 0960-894X, 4 p.Article

A novel convergent method for the synthesis of α-acyl-γ-hydroxylactams and its application in the total synthesis of PI-090 and 091UCHIRO, Hiromi; SHIONOZAKI, Nobuhiro; KOBAYAKAWA, Yu et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 14, pp 4765-4768, issn 0960-894X, 4 p.Article

A novel series of G-quadruplex ligands with selectivity for HIF-expressing osteosarcoma and renal cancer cell linesLOMBARDO, Caterina M; WELSH, Sarah J; STRAUSS, Sandra J et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 18, pp 5984-5988, issn 0960-894X, 5 p.Article

A σ₁ receptor pharmacophore derived from a series of N-substituted 4-azahexacyclo[5.4.1.0^2,6.0^3,10.0^5,9.0^8,11]dodecan-3-ols (AHDs)BANISTER, Samuel D; MANOLI, Miral; REDDY DODDAREDDY, Munikumar et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 19, pp 6053-6058, issn 0960-894X, 6 p.Article

Activation of human RNase L by 2'- and 5'-O-methylphosphonate-modified oligoadenylatesPAV, Ondřej; PANOVA, Natalya; SNASEL, Jan et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 1, pp 181-185, issn 0960-894X, 5 p.Article

Activity-based fluorescent probes for monitoring sulfatase activityPARK, Hyun-Joo; RHEE, Hyun-Woo; HONG, Jong-In et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 15, pp 4939-4941, issn 0960-894X, 3 p.Article

Aminopyrimidinone Cdc7 Kinase InhibitorsWOODS, Keith W; LAI, Chunqiu; JOHNSON, Eric F et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 5, pp 1940-1943, issn 0960-894X, 4 p.Article

An approach for differentiating isozymes. Construction of libraries containing short aromatic peptides as part of a method to design selective inhibitors against lipasesPARK, Sangeun; YU, Jaehoon.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 9, pp 3147-3151, issn 0960-894X, 5 p.Article

An efficient one-pot synthesis and photoinduced DNA cleavage studies of 2-chloro-3-(5-aryl-4,5-dihydroisoxazol-3-yl)quinolinesBINDU, P. J; MAHADEVAN, K. M; RAVIKUMAR NAIK, T. R et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 19, pp 6095-6098, issn 0960-894X, 4 p.Article

Anion-selective transport activities of tetrameric sterol―spermine conjugatesCHEN, Wen-Hua; JIA ZHOU; WANG, Yong-Min et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 12, pp 4010-4013, issn 0960-894X, 4 p.Article

Antagonists of 5-HT6 receptors. Substituted 3-(phenylsulfonyl) pyrazolo[1,5-a]pyrido[3,4-e]pyrimidines and 3-(phenylsulfonyl) pyrazolo[1,5-a]pyrido[4,3-d]pyrimidines―Synthesis and 'structure―activity' relationshipIVACHTCHENKO, Alexandre V; GOLOVINA, Elena S; KADIEVA, Madina G et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 13, pp 4273-4280, issn 0960-894X, 8 p.Article

Anti-inflammatory sesquiterpene lactones from the flower of Vernonia cinereaUI JOUNG YOUN; PARK, Eun-Jung; LENG CHEE CHANG et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 17, pp 5559-5562, issn 0960-894X, 4 p.Article

Anti-tumor activity of new orally bioavailable 2-amino-5-(thiophen-2-yl) benzamide-series histone deacetylase inhibitors, possessing an aqueous soluble functional group as a surface recognition domainHIRATA, Yoshiyuki; HIRATA, Masahiko; KAWARATANI, Yasuyuki et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 5, pp 1926-1930, issn 0960-894X, 5 p.Article

Assay and inhibition of diacylglycerol lipase activityJOHNSTON, Meghan; BHATT, Shachi R; SIKKA, Surina et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 14, pp 4585-4592, issn 0960-894X, 8 p.Article

Benzoylbenzimidazole-based selective inhibitors targeting Cryptosporidium parvum and Toxoplasma gondii calcium-dependent protein kinase-1ZHONGSHENG ZHANG; OJO, Kayode K; MALY, Dustin J et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 16, pp 5264-5267, issn 0960-894X, 4 p.Article

Bio-inspired synthesis and biological evaluation of a colchicine-related compound libraryNICOLAOU, K. C; VALIULIN, Roman A; POKORSKI, Jonathan K et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 11, pp 3776-3780, issn 0960-894X, 5 p.Article