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Stereoselective Halofantrine and desbutylhalofantrine disposition in the rat: Cardiac and plasma concentrations and plasma protein binding

Author
BROCKS, Dion R1
[1] Faculty of Pharmacy and Pharmaceutical Sciences, University of Alberta, Edmonton, AB, T6G 2N8, Canada
Source

Biopharmaceutics & drug disposition. 2002, Vol 23, Num 1, pp 9-15 ; ref : 17 ref

CODEN
BDDID8
ISSN
0142-2782
Scientific domain
Pharmacology drugs
Publisher
Wiley, Chichester
Publication country
United Kingdom
Document type
Article
Language
English
Keyword (fr)
Animal Antipaludique Capacité fixation Chimiothérapie Coeur Distribution Enantiomère Halofantrine Métabolite Pharmacocinétique Plasma sanguin Protéine Racémique Rat Stéréoisomère Stéréosélectivité Toxicité Traitement Trouble rythme cardiaque Voie intraveineuse Appareil circulatoire pathologie Mammalia Rodentia Vertebrata
Keyword (en)
Animal Antimalarial Binding capacity Chemotherapy Heart Distribution Enantiomer Halofantrine Metabolite Pharmacokinetics Blood plasma Protein Racemic Rat Stereoisomer Stereoselectivity Toxicity Treatment Arrhythmia Intravenous administration Cardiovascular disease Mammalia Rodentia Vertebrata
Keyword (es)
Animal Antipalúdico Capacidad de fijación Quimioterapia Corazón Distribución Enantiómero Halofantrina Metabolito Farmacocinética Plasma sanguíneo Proteína Racémico Rata Estereoisómero Estereoselectividad Toxicidad Tratamiento Arritmia Vía intravenosa Aparato circulatorio patología Mammalia Rodentia Vertebrata
Classification
Pascal
002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02U Drug toxicity and drugs side effects treatment / 002B02U03 Toxicity: cardiovascular system

Discipline
Drugs toxicity and drug intoxications Toxicology
Origin
Inist-CNRS
Database
PASCAL
INIST identifier
13550068

Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS

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