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AH-1058: A novel cardioselective Ca2+ channel blocker

Author
TAKAHARA, Akira1 ; SUGIYAMA, Atsushi2 ; YOSHIMOTO, Ryota1 ; HASHIMOTO, Keitaro2
[1] Pharmaceutical Research Laboratories, Ajinomoto Co., Inc., Kawasaki, Japan
[2] Department of Pharmacology, Yamanashi Medical University, Yamanashi, Japan
Source

Cardiovascular drug reviews (Print). 2001, Vol 19, Num 4, pp 279-296 ; ref : 48 ref

CODEN
CDREEA
ISSN
0897-5957
Scientific domain
Cardiology, blood circulation, phlebology; Pharmacology drugs
Publisher
Blackwell, Malden, MA
Publication country
United States
Document type
Article
Language
English
Keyword (fr)
Activité biologique Animal Antagoniste calcium Antiarythmique Antihistaminique Appareil circulatoire Calcium Canal ionique Chien Cobaye Coeur Cyproheptadine In vitro In vivo Muscle lisse Myocarde Myocyte Mécanisme action Rat Relation structure activité Relâchement musculaire Récepteur histaminergique H1 Vasodilatateur Voie intraveineuse AH 1058 Carnivora Fissipedia Mammalia Rodentia Vertebrata
Keyword (en)
Biological activity Animal Calcium antagonist Antiarrhythmic agent Antihistaminic Circulatory system Calcium Ionic channel Dog Guinea pig Heart Cyproheptadine In vitro In vivo Smooth muscle Myocardium Myocyte Mechanism of action Rat Structure activity relation Muscular relaxation H1 Histamine receptor Vasodilator agent Intravenous administration Carnivora Fissipedia Mammalia Rodentia Vertebrata
Keyword (es)
Actividad biológica Animal Antagonista calcio Antiarrítmico Antihistamínico Aparato circulatorio Calcio Canal iónico Perro Cobayo Corazón Ciproheptadina In vitro In vivo Músculo liso Miocardio Miocito Mecanismo acción Rata Relación estructura actividad Relajación muscular Receptor histaminérgico H1 Vasodilatador Vía intravenosa Carnivora Fissipedia Mammalia Rodentia Vertebrata
Classification
Pascal
002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02F Cardiovascular system / 002B02F02 Antiarythmic agents

Pascal
002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02F Cardiovascular system / 002B02F09 Miscellaneous

Discipline
Pharmacological treatments
Origin
Inist-CNRS
Database
PASCAL
INIST identifier
13589372

Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS

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