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The mechanism of the irreversible inhibition of estrone sulfatase (ES) through the consideration of a range of methane- and amino-sulfonate-based compounds

Author
AHMED, Sabbir1 ; JAMES, Karen2 ; OWEN, Caroline P1 ; PATELA, Chirag K1 ; SAMPSON, Luther3
[1] School of Chemical and Pharmaceutical Sciences, Kingston University, Penrhyn Road, Kingston upon Thames, Surrey, KT1 2EE, United Kingdom
[2] Institute of Cancer Research, Sutton, United Kingdom
[3] Novartis Pharma AG, 4002 Basel, Switzerland
Source

Bioorganic & medicinal chemistry letters (Print). 2002, Vol 12, Num 9, pp 1279-1282

ISSN
0960-894X
Scientific domain
Biochemistry, molecular biology, biophysics; Pharmacology drugs
Publisher
Elsevier, Oxford
Publication country
United Kingdom
Document type
Article
Language
English
Keyword (fr)
Amidosulfate organique Arylsulfatase Benzène dérivé Composé aliphatique Composé non stéroïde Inhibiteur enzyme Mécanisme action Relation structure activité Réaction irréversible Steryl-sulfatase Estrone sulfatase Enzyme Esterases Hydrolases Sulfuric ester hydrolases
Keyword (en)
Organic amidosulfate Arylsulfatase Benzene derivatives Aliphatic compound Non steroid compound Enzyme inhibitor Mechanism of action Structure activity relation Irreversible reaction Steryl-sulfatase Enzyme Esterases Hydrolases Sulfuric ester hydrolases
Keyword (es)
Amidosulfato orgánico Arylsulfatase Benceno derivado Compuesto alifático Compuesto no esteroide Inhibidor enzima Mecanismo acción Relación estructura actividad Reacción irreversible Steryl-sulfatase Enzima Esterases Hydrolases Sulfuric ester hydrolases
Classification
Pascal
002 Biological and medical sciences / 002A Fundamental and applied biological sciences. Psychology / 002A02 Analytical, structural and metabolic biochemistry / 002A02E Enzymes and enzyme inhibitors / 002A02E04 Hydrolases

Pascal
002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02W Miscellaneous

Discipline
Analytical, structural and metabolic biochemistry General pharmacology
Origin
Inist-CNRS
Database
PASCAL
INIST identifier
13610174

Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS

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