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The novel and systemically active metabotropic glutamate 1 (mGlu1) receptor antagonist 3-MATIDA reduces post-ischemic neuronal death

Author
MORONI, Flavio1 ; ATTUCCI, Sabina1 ; COZZI, Andrea1 ; MELI, Elena1 ; PICCA, Roberta1 ; SCHEIDELER, Mark A2 ; PELLICCIARI, Roberto3 ; NOE, Christian4 ; SARICHELOU, Iran2 ; PELLEGRINI-GIAMPIETRO, Domenico E1
[1] Dipartimento di Farmacologia Preclinica e Clinica, Università di Firenze, Viale Pieraccini 6, 50139 Firenze, Italy
[2] GlaxoSmithKline Pharmaceuticals, Neurobiology Research, Via Zambeletti, 20021 Baranzate di Bollate (Milano), Italy
[3] Dipartimento di Chimica e Tecnologia del Farmaco, Università di Perugia, Via del Liceo 1, 06127 Perugia, Italy
[4] Institute of Pharmaceutical Chemistry, University of Vienna, Althanstrasse 14, 1090 Vienna, Austria
Source

Neuropharmacology. 2002, Vol 42, Num 6, pp 741-751 ; ref : 1 p.1/2

CODEN
NEPHBW
ISSN
0028-3908
Scientific domain
Neurology; Pharmacology drugs; Psychology, psychopathology, psychiatry
Publisher
Elsevier, Oxford
Publication country
United Kingdom
Document type
Article
Language
English
Keyword (fr)
Activité biologique Agoniste Animal nouveau né Antagoniste Appareil circulatoire pathologie Appareil urinaire Chimiothérapie Encéphale pathologie Encéphale Hamster In vitro In vivo Mécanisme action Neuroprotecteur Prévention Rat Rein Récepteur glutamate mglu groupe I Récepteur glutamate Récepteur métabotropique Système nerveux central Transfection Mammalia Rodentia Système nerveux central pathologie Système nerveux pathologie Vertebrata
Keyword (en)
Biological activity Agonist Newborn animal Antagonist Cardiovascular disease Urinary system Chemotherapy Cerebral disorder Brain (vertebrata) Hamster In vitro In vivo Mechanism of action Neuroprotective agent Prevention Rat Kidney Group I mglu glutamate receptor Glutamate receptor Metabotropic receptor Central nervous system Transfection Mammalia Rodentia Central nervous system disease Nervous system diseases Vertebrata
Keyword (es)
Actividad biológica Agonista Animal recién nacido Antagonista Aparato circulatorio patología Aparato urinario Quimioterapia Encéfalo patología Encéfalo Hamster In vitro In vivo Mecanismo acción Neuroprotector Prevención Rata Riñón Réceptor glutamato grupo I Receptor glutámato Receptor metabotropico Sistema nervioso central Transfección Mammalia Rodentia Sistema nervosio central patología Sistema nervioso patología Vertebrata
Classification
Pascal
002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02B Neuropharmacology / 002B02B09 Neurotransmitters. Neurotransmission. Receptors / 002B02B09E Glutamatergic system (aspartate and other excitatory aminoacids)

Pascal
002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02B Neuropharmacology / 002B02B10 Neuroprotective agent

Discipline
Pharmacological treatments
Origin
Inist-CNRS
Database
PASCAL
INIST identifier
13672452

Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS

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