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The pharmacokinetics of sumatriptan when administered with clarithromycin in healthy volunteers

Author
MOORE, Katy H. P1 ; LEESE, Philip T2 ; MCNEAL, Scott1 ; GRAY, Peter2 ; O'QUINN, Stephen1 ; BYE, Carole3 ; SALE, Mark1
[1] GlaxoSmithKline, Research Triangle Park, North Carolina, United States
[2] Quintiles, Lenexa, Kansas, United States
[3] GlaxoSmithKline, Greenford, Middlesex, United Kingdom
Source

Clinical therapeutics. 2002, Vol 24, Num 4, pp 583-594 ; ref : 25 ref

ISSN
0149-2918
Scientific domain
Pharmacology drugs
Publisher
Excerpta Medica, Belle Mead, NJ
Publication country
United States
Document type
Article
Language
English
Keyword (fr)
Agoniste Amine oxidase (flavin-containing) Antibactérien Antibiotique Antimigraineux Association médicamenteuse Chimiothérapie Clarithromycine Cytochrome P450 Homme Individu sain Interaction médicamenteuse Macrolide Métabolisme Pharmacocinétique Plasma sanguin Récepteur sérotoninergique Stimulant sérotoninergique Sumatriptan Traitement Voie orale Volontaire Cytochrome CYP3A4 Enzyme Oxidoreductases
Keyword (en)
Agonist Amine oxidase (flavin-containing) Antibacterial agent Antibiotic Antimigrainous agent Drug combination Chemotherapy Clarithromycin Cytochrome P450 Human Healthy subject Drug interaction Macrolide Metabolism Pharmacokinetics Blood plasma Serotonine receptor Serotonin agonist Sumatriptan Treatment Oral administration Volunteer Enzyme Oxidoreductases
Keyword (es)
Agonista Amine oxidase (flavin-containing) Antibacteriano Antibiótico Agente antimigrañoso Asociación medicamentosa Quimioterapia Claritromicina Citocromo P450 Hombre Individuo sano Interacción medicamentosa Macrólido Metabolismo Farmacocinética Plasma sanguíneo Receptor serotoninérgico Estimulante serotoninérgico Sumatriptán Tratamiento Vía oral Voluntario Enzima Oxidoreductases
Classification
Pascal
002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02A General pharmacology / 002B02A05 Pharmacokinetics. Pharmacogenetics. Drug-receptor interactions

Discipline
General pharmacology
Origin
Inist-CNRS
Database
PASCAL
INIST identifier
14186647

Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS

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