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Presystemic metabolism and intestinal absorption of antipsoriatic fumaric acid esters

Author
WERDENBERG, D1 ; JOSHI, R2 ; WOLFFRAM, S3 ; MERKLE, H. P1 ; LANGGUTH, P4
[1] Department of Applied Biosciences, Swiss Federal Institute of Technology Zurich, Winterthurerstrasse 190, 8057 Zurich, Switzerland
[2] Fumapharm AG, 5630 Muri, Switzerland
[3] Institute of Animal Nutrition, Physiology and Metabolism, Christian-Albrechts-University of Kiel, 24098 Kiel, Germany
[4] Department of Biopharmaceutics and Pharmaceutical Technology, Johannes Gutenberg-University, 55099 Mainz, Germany
Source

Biopharmaceutics & drug disposition. 2003, Vol 24, Num 6, pp 259-273, 15 p ; ref : 54 ref

CODEN
BDDID8
ISSN
0142-2782
Scientific domain
Pharmacology drugs
Publisher
Wiley, Chichester
Publication country
United Kingdom
Document type
Article
Language
English
Author keyword
bioavailability degradation first-pass extraction permeability prodrug
Keyword (fr)
Absorption Analogue Animal Antipsoriasique Biodisponibilité Dégradation Ester Fumarique acide In vitro Intestin Métabolisme Perméabilité Promédicament
Keyword (en)
Absorption Analog Animal Antipsoriatic agent Bioavailability Degradation Ester Fumaric acid In vitro Gut Metabolism Permeability Prodrug
Keyword (es)
Absorción Análogo Animal Antipsoriásico Biodisponibilidad Degradación Ester Fumarico ácido In vitro Intestino Metabolismo Permeabilidad Promedicamento
Classification
Pascal
002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02K Skin, nail, hair, dermoskeleton

Discipline
Pharmacological treatments
Origin
Inist-CNRS
Database
PASCAL
INIST identifier
15101482

Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS

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