Synthesis and evaluation of aminophosphinic acid derivatives as inhibitors of renal dipeptidase
- Author
- GURULINGAPPA, Hallur1 ; BUCKHALTS, Phillip1 ; KINZLER, Kenneth W1 ; VOGELSTEIN, Bert1 ; KHAN, Saeed R1
[1] The Sidney Kimmel Comprehensive Cancer Center at Johns Hopkins, Baltimore, MD 21231, United States - Source
Bioorganic & medicinal chemistry letters (Print). 2004, Vol 14, Num 13, pp 3531-3533, 3 p
- ISSN
- 0960-894X
- Scientific domain
- Biochemistry, molecular biology, biophysics; Pharmacology drugs
- Publisher
- Elsevier, Oxford
- Publication country
- United Kingdom
- Document type
- Article
- Language
- English
- Keyword (fr)
- Aminoacide Benzène dérivé Cyclohexane dérivé In vitro Inhibiteur enzyme Membrane dipeptidase Phosphinique acide Relation structure activité Synthèse chimique Benzèneacrylique acide dérivé Dipeptidases Enzyme Halogène Composé organique Hydrolases Peptidases Phosphore Composé organique
- Keyword (en)
- Aminoacid Benzene derivatives Cyclohexane derivatives In vitro Enzyme inhibitor Membrane dipeptidase Phosphinic acids Structure activity relation Chemical synthesis Dipeptidases Enzyme Halogen Organic compounds Hydrolases Peptidases Phosphorus Organic compounds
- Keyword (es)
- Aminoácido Benceno derivado Ciclohexano derivado In vitro Inhibidor enzima Membrane dipeptidase Relación estructura actividad Síntesis química Dipeptidases Enzima Halógeno Compuesto orgánico Hydrolases Peptidases Fósforo Compuesto orgánico
- Classification
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02W Miscellaneous
- Discipline
- General pharmacology
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 15797321
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1016/j.bmcl.2004.04.057 
https://dx.doi.org/10.1016/j.bmcl.2004.04.057
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