Synthesis of a bromotyrosine-derived natural product inhibitor of mycothiol-s-conjugate amidase
- Author
- FETTEROLF, Brandon1 ; BEWLEY, Carole A1
[1] Laboratory of Bioorganic Chemistry, National Institute of Diabetes and Digestive and Kidney Diseases, National Institutes of Health, Bethesda, MD 20892-0820, United States - Source
Bioorganic & medicinal chemistry letters (Print). 2004, Vol 14, Num 14, pp 3785-3788, 4 p ; ref : 22 ref
- ISSN
- 0960-894X
- Scientific domain
- Biochemistry, molecular biology, biophysics; Pharmacology drugs
- Publisher
- Elsevier, Oxford
- Publication country
- United Kingdom
- Document type
- Article
- Language
- English
- Keyword (fr)
- Alcaloïde Amidase Composé conjugué Détoxication In vitro Inhibiteur enzyme Mycobacterium tuberculosis Oxime Relation structure activité Synthèse chimique Synthèse totale α-Aminoacide Agmatine dérivé Mycothiol-S-conjugate amidase Tyrosine dérivé Actinomycetes Bactérie Brome Composé organique Enzyme Hydrolases Mycobacteriaceae Mycobacteriales
- Keyword (en)
- Alkaloid Amidase Conjugated compound Detoxification In vitro Enzyme inhibitor Mycobacterium tuberculosis Oxime Structure activity relation Chemical synthesis Total synthesis α-Aminoacid Actinomycetes Bacteria Bromine Organic compounds Enzyme Hydrolases Mycobacteriaceae Mycobacteriales
- Keyword (es)
- Alcaloide Amidase Compuesto conjugado Detoxicación In vitro Inhibidor enzima Mycobacterium tuberculosis Oxima Relación estructura actividad Síntesis química Síntesis total α-Aminoácido Actinomycetes Bacteria Bromo Compuesto orgánico Enzima Hydrolases Mycobacteriaceae Mycobacteriales
- Classification
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02W Miscellaneous
- Discipline
- General pharmacology
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 15889630
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1016/j.bmcl.2004.04.095 
https://dx.doi.org/10.1016/j.bmcl.2004.04.095
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