Novel azapeptide inhibitors of hepatitis C virus serine protease
- Author
- BAILEY, Murray D1 ; HALMOS, Ted1 ; GOUDREAU, Nathalie1 ; LESCOP, Ewen1 ; LLINAS-BRUNET, Montse1
[1] Boehringer Ingelheim (Canada) Ltd. Research and Development, 2100 Canard Street, Laval, Quebec H7S 2G5, Canada - Source
Journal of medicinal chemistry (Print). 2004, Vol 47, Num 15, pp 3788-3799, 12 p ; ref : 35 ref
- CODEN
- JMCMAR
- ISSN
- 0022-2623
- Scientific domain
- Pharmacology drugs
- Publisher
- American Chemical Society, Washington, DC
- Publication country
- United States
- Document type
- Article
- Language
- English
- Keyword (fr)
- Antiviral Carbazate organique In vitro Inhibiteur enzyme Peptide Pseudopeptide Relation structure activité Serine endopeptidases Synthèse chimique Virus hépatite C Azapeptide Enzyme Flaviviridae Hepacivirus Hydrolases Peptidases Virus
- Keyword (en)
- Antiviral Organic carbazate In vitro Enzyme inhibitor Peptides Pseudopeptide Structure activity relation Serine endopeptidases Chemical synthesis Hepatitis C virus Enzyme Flaviviridae Hepacivirus Hydrolases Peptidases Virus
- Keyword (es)
- Antiviral Carbazato orgánico In vitro Inhibidor enzima Péptido Seudopéptido Relación estructura actividad Serine endopeptidases Síntesis química Hepatitis C virus Enzima Flaviviridae Hepacivirus Hydrolases Peptidases Virus
- Classification
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02S Antibiotics. Antiinfectious agents. Antiparasitic agents / 002B02S05 Antiviral agents
- Discipline
- Pharmacological treatments
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 15940088
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1021/jm049864b 
https://dx.doi.org/10.1021/jm049864b
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