Novel glycine transporter type-2 reuptake inhibitors. Part 1: α-amino acid derivatives
- Author
- WOLIN, Ronald L1 ; VENKATESAN, Hariharan1 ; LIU TANG1 ; SANTILLAN, Alejandro JR1 ; BARCLAY, Tristin1 ; WILSON, Sandy1 ; DOO HYUN LEE1 ; LOVENBERG, Timothy W1
[1] Johnson & Johnson Pharmaceutical Research and Development, LLC, 3210, Merryfield Row, San Diego, CA 92121, United States - Source
Bioorganic & medicinal chemistry. 2004, Vol 12, Num 16, pp 4477-4492, 16 p ; ref : 19 ref
- ISSN
- 0968-0896
- Scientific domain
- Biochemistry, molecular biology, biophysics; Pharmacology drugs
- Publisher
- Elsevier Science, Oxford
- Publication country
- United Kingdom
- Document type
- Article
- Language
- English
- Keyword (fr)
- Amine Aminoamide Benzène dérivé Biphényle dérivé Glycine Homme In vitro Inhibiteur recapture Inhibition Relation structure activité Synthèse chimique Transport biologique Urées α-Aminoacide Phénylalaninamide dérivé Transporteur glycine GLYT2
- Keyword (en)
- Amine Aminoamide Benzene derivatives Biphenyl derivatives Glycine Human In vitro Reuptake inhibitor Inhibition Structure activity relation Chemical synthesis Biological transport Ureas α-Aminoacid GLYT2 glycine transporter
- Keyword (es)
- Amina Aminoamida Benceno derivado Bifenilo derivado Glicina Hombre In vitro Inhibidor recaptura Inhibición Relación estructura actividad Síntesis química Transporte biológico Ureas α-Aminoácido
- Classification
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02B Neuropharmacology / 002B02B09 Neurotransmitters. Neurotransmission. Receptors / 002B02B09G Miscellaneous
- Discipline
- Pharmacological treatments
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 15973892
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1016/j.bmc.2004.05.042 
https://dx.doi.org/10.1016/j.bmc.2004.05.042
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