Synthesis and evaluation of 2-amino-8-alkoxy quinolines as MCHr1 antagonists. Part 1
- Author
- SOUERS, Andrew J1 ; WODKA, Dariusz1 ; HERNANDEZ, Lisa E1 ; MARSH, Kennan C1 ; COLLINS, Christine A1 ; KYM, Philip R1 ; JU GAO1 ; LEWIS, Jared C1 ; VASUDEVAN, Anil1 ; GENTLES, Robert1 ; BRODJIAN, Sevan1 ; DAYTON, Brian1 ; OGIELA, Christopher A1 ; FRY, Dennis1
[1] Metabolic Diseases Research, Global Pharmaceutical Research and Development, Abbott Laboratories, Abbott Park, IL 60064, United States - Source
Bioorganic & medicinal chemistry letters (Print). 2004, Vol 14, Num 19, pp 4873-4877, 5 p
- ISSN
- 0960-894X
- Scientific domain
- Biochemistry, molecular biology, biophysics; Pharmacology drugs
- Publisher
- Elsevier, Oxford
- Publication country
- United Kingdom
- Document type
- Article
- Language
- English
- Keyword (fr)
- Animal Antagoniste Automatisation Chimie combinatoire Criblage Hormone concentrant mélanine Pharmacocinétique Quinoléine dérivé Relation structure activité Récepteur biologique Souris Synthèse chimique Voie orale Mammalia Rodentia Vertebrata
- Keyword (en)
- Animal Antagonist Automation Combinatorial chemistry Screening Melanin concentrating hormone Pharmacokinetics Quinoline derivatives Structure activity relation Biological receptor Mouse Chemical synthesis Oral administration Mammalia Rodentia Vertebrata
- Keyword (es)
- Animal Antagonista Automatización Química combinatoria Cernido Hormona concentración melanina Farmacocinética Quinolina derivado Relación estructura actividad Receptor biológico Ratón Síntesis química Vía oral Mammalia Rodentia Vertebrata
- Classification
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02W Miscellaneous
- Discipline
- General pharmacology
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 16101734
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1016/j.bmcl.2004.07.032 
https://dx.doi.org/10.1016/j.bmcl.2004.07.032
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