Synthesis and evaluation of 4-triazolylflavans as new aromatase inhibitors
- Author
- YAHIAOUI, Samir1 ; POUGET, Christelle1 ; FAGNERE, Catherine1 ; CHAMPAVIER, Yves2 ; HABRIOUX, Gérard1 ; CHULIA, Albert José1
[1] UPRES EA 1085 ' Biomolécules et Cibles Cellulaires Tumorales, ' Faculté de Pharmacie. 2 rue du Docteur Marcland, 87025 Limoges, France
[2] Service Commun de RMN de l'Université de Limoges, Faculté de Pharmacie, 2 rue du Docteur Marcland, 87025 Limoges, France - Source
Bioorganic & medicinal chemistry letters (Print). 2004, Vol 14, Num 20, pp 5215-5218, 4 p ; ref : 18 ref
- ISSN
- 0960-894X
- Scientific domain
- Biochemistry, molecular biology, biophysics; Pharmacology drugs
- Publisher
- Elsevier, Oxford
- Publication country
- United Kingdom
- Document type
- Article
- Language
- English
- Keyword (fr)
- Activité biologique Anastrozole Anticancéreux Estrogen synthase Flavonoïde Glande mammaire Inhibiteur enzyme Inhibition Létrozole Synthèse chimique Traitement Triazole dérivé Tumeur Flavane dérivé Enzyme
- Keyword (en)
- Biological activity Anastrozole Antineoplastic agent Estrogen synthase Flavonoid Mammary gland Enzyme inhibitor Inhibition Letrozole Chemical synthesis Treatment Triazole derivatives Tumor Enzyme
- Keyword (es)
- Actividad biológica Anastrozol Anticanceroso Estrogen synthase Flavonoide Glándula mamaria Inhibidor enzima Inhibición Letrozol Síntesis química Tratamiento Triazol derivado Tumor Enzima
- Classification
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02R Antineoplastic agents / 002B02R01 General aspects
- Discipline
- Pharmacological treatments
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 16119678
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1016/j.bmcl.2004.07.090 
https://dx.doi.org/10.1016/j.bmcl.2004.07.090
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