Synthesis of 1,4-benzodiazepine-3,5-diones
- Author
- WIKLUND, Per1 ; ROGERS-EVANS, Mark2 ; BERGMAN, Jan1
[1] Unit for Organic Chemistry, Department of Biosciences, Karolinska Institute and Södertörn University College, Novum Research Park, 141 57 Huddinge, Sweden
[2] F. Hoffmann-La Roche Ltd, Pharmaceuticals Division, Lead Generation, PRBC-CI, Bldg 65/416, 4070 Basel, Switzerland - Source
Journal of organic chemistry. 2004, Vol 69, Num 19, pp 6371-6376, 6 p
- CODEN
- JOCEAH
- ISSN
- 0022-3263
- Scientific domain
- Biochemistry, molecular biology, biophysics; Organic chemistry
- Publisher
- American Chemical Society, Washington, DC
- Publication country
- United States
- Document type
- Article
- Language
- English
- Keyword (fr)
- Anthranilique acide Benzodiazépine dérivé Caractérisation Carboxamide Composé aromatique Composé nitroso Contraction cycle Cyclisation Dicétone Dénitrosation Effet substituant Ester Hétérocycle azote Mécanisme réaction Quinazoline dérivé Synthèse chimique Transposition chimique 1,4-Benzodiazépine-3,5-dione dérivé
- Keyword (en)
- Anthranilic acid Benzodiazepine derivatives Characterization Carboxamide Aromatic compound Nitroso compound Ring contraction Cyclization Diketone Denitrosation Substituent effect Ester Nitrogen heterocycle Reaction mechanism Quinazoline derivatives Chemical synthesis Chemical rearrangement
- Keyword (es)
- Anthranilic acid Benzodiazepina derivado Caracterización Carboxamida Compuesto aromático Compuesto nitroso Contracción ciclo Ciclización Dicetona Desnitrosación Efecto sustituyente Ester Heterociclo nitrógeno Mecanismo reacción Síntesis química Transposición química
- Classification
- Pascal
- 001 Exact sciences and technology / 001C Chemistry / 001C03 Organic chemistry / 001C03C Preparations and properties / 001C03C06 Heterocyclic compounds / 001C03C06C Heterocyclic compounds with several n hetero atoms in the same ring, in separated rings or in fused rings
- Discipline
- Organic chemistry
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 16123490
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1021/jo049169b 
https://dx.doi.org/10.1021/jo049169b
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