New COOX-2/5-LOX inhibitors: Apoptosis-inducing agents potentially useful in prostate cancer chemotherapy
- Author
- POMMERY, Nicole; TAVERNE, Thierry; TELLIEZ, Aurélie; GOOSSENS, Laurence; CHARLIER, Caroline; POMMERY, Jean; GOOSSENS, Jean-Francois; HOUSSIN, Raymond; DURANT, Francois; HENICHART, Jean-Pierre
Institut de Chimie Pharmaceutique Albert Lespagnol, EA 2692, Université de Lille 2, BP 83, 59006 Lille, France
Laboratoire de Chimie Moléculaire Structurale, Facultés Universitaires Notre-Dame de la Paix, rue de Bruxelles, 5000 Namur, Belgium - Source
Journal of medicinal chemistry (Print). 2004, Vol 47, Num 25, pp 6195-6206, 12 p ; ref : 43 ref
- CODEN
- JMCMAR
- ISSN
- 0022-2623
- Scientific domain
- Pharmacology drugs
- Publisher
- American Chemical Society, Washington, DC
- Publication country
- United States
- Document type
- Article
- Language
- English
- Keyword (fr)
- Activité biologique Anticancéreux Apoptose Chimiothérapie Composé benzénique Cyclooxygenase 2 Ether Fluor composé organique In vitro Inhibiteur enzyme Modèle moléculaire Modélisation Oxidoreductases Prostate Pyrane dérivé Pyrazole dérivé Sulfonamide Synthèse chimique Tumeur 5-Lipoxygenase Benzènesulfonamide(4-[3-(3-fluoro-5-[4-méthoxy-tétrahydropyran-4-yl]phénoxyméthyl)-5-phénylpyrazol-1-yl]) Enzyme
- Keyword (en)
- Biological activity Antineoplastic agent Apoptosis Chemotherapy Benzenic compound Cyclooxygenase 2 Ether Organic fluorine compounds In vitro Enzyme inhibitor Molecular model Modeling Oxidoreductases Prostate Pyran derivatives Pyrazole derivatives Sulfonamide Chemical synthesis Tumor Enzyme
- Keyword (es)
- Actividad biológica Anticanceroso Apoptosis Quimioterapia Compuesto bencénico Cyclooxygenase 2 Eter In vitro Inhibidor enzima Modelo molecular Modelización Oxidoreductases Prostata Pirano derivado Pirazol derivado Sulfonamida Síntesis química Tumor Enzima
- Classification
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02R Antineoplastic agents / 002B02R01 General aspects
- Discipline
- Pharmacological treatments
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 16305158
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1021/jm0407761 
https://dx.doi.org/10.1021/jm0407761
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