Non-imidazole histamine H3 ligands. Part III. New 4-n-propylpiperazines as non-imidazole histamine H3-antagonists
- Author
- WALCZYNSKI, Krzysztof1 ; ZUIDERVELD, Obbe P2 ; TIMMERMAN, Henk2
[1] Department of Synthesis and Technology of Drugs, Medical University Muszyńskiego, MuszyńskiegoStreet 1, 90-145 Łódź, Poland
[2] Leiden/Amsterdam Centre for Drug Research, Division of Medicinal Chemistry, Vrije Universiteit, De Boelelaan 1083, 1081 HV Amsterdam, Netherlands - Source
European journal of medicinal chemistry. 2005, Vol 40, Num 1, pp 15-23, 9 p ; ref : 50 ref
- CODEN
- EJMCA5
- ISSN
- 0223-5234
- Scientific domain
- Organic chemistry; Pharmacology drugs
- Publisher
- Elsevier, Oxford
- Publication country
- United Kingdom
- Document type
- Article
- Language
- English
- Author keyword
- 1-[(2- Benzothiazole)-4-n-propyl]piperazine 1-[(2-Benzooxazole)-4-n-propyl]piperazine 1-[(2-Thiazolopyridine)-4-n-propyl]piperazines;1[(2-Oxazolopyridine)-4-n-propyl]piperazines H3-antagonists Histamine H3-receptor
- Keyword (fr)
- Animal Antagoniste Benzooxazole dérivé Benzothiazole dérivé Cobaye In vitro Pipérazine dérivé Relation structure activité Récepteur histaminergique H3 Synthèse chimique Oxazolopyridine Thiazolo[4,5-b]pyridine dérivé Thiazolo[4,5-c]pyridine(2-[4-propylpipérazino]) Thiazolo[5,4-b]pyridine dérivé Thiazolopyridine Mammalia Rodentia Vertebrata
- Keyword (en)
- Animal Antagonist Benzoxazole derivatives Benzothiazole derivatives Guinea pig In vitro Piperazine derivatives Structure activity relation H3 histamine receptor Chemical synthesis Mammalia Rodentia Vertebrata
- Keyword (es)
- Animal Antagonista Benzotiazol derivado Cobayo In vitro Piperazina derivado Relación estructura actividad Receptor histaminérgico H3 Síntesis química Mammalia Rodentia Vertebrata
- Classification
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02B Neuropharmacology / 002B02B09 Neurotransmitters. Neurotransmission. Receptors / 002B02B09G Miscellaneous
- Discipline
- Pharmacological treatments
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 16446832
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1016/j.ejmech.2004.09.010 
https://dx.doi.org/10.1016/j.ejmech.2004.09.010
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