Non-peptidic small molecule inhibitors of XIAP
- Author
- PARK, Cheol-Min1 ; CHAOHONG SUN2 ; OLEJNICZAK, Edward T2 ; WILSON, Alan E1 ; MEADOWS, Robert P2 ; BETZ, Stephen F2 ; ELMORE, Steven W1 ; FESIK, Stephen W1
[1] Cancer Research, Global Pharmaceutical R&D, Abbott Laboratories, 100 Abbott Park Rd, Abbott Park, IL 60064-6010, United States
[2] Advanced Technology, Global Pharmaceutical R&D, Abbott Laboratories, 100 Abbott Park Rd, Abbott Park, IL 60064-6010, United States - Source
Bioorganic & medicinal chemistry letters (Print). 2005, Vol 15, Num 3, pp 771-775, 5 p
- ISSN
- 0960-894X
- Scientific domain
- Biochemistry, molecular biology, biophysics; Pharmacology drugs
- Publisher
- Elsevier, Oxford
- Publication country
- United Kingdom
- Document type
- Article
- Language
- English
- Keyword (fr)
- Anticancéreux Apoptose Composé non peptide Imidazole dérivé In vitro Inhibiteur Mimétique Relation structure activité Synthèse chimique Thiazole dérivé Protéine SMAC Protéine inhibition apoptose Thiazole(2-alanylamino-4-[4-bromophényl]-5-phényl)
- Keyword (en)
- Antineoplastic agent Apoptosis Non peptide compound Imidazole derivatives In vitro Inhibitor Mimetic Structure activity relation Chemical synthesis Thiazole derivatives Second mitochondria derived activator of caspase protein Apoptosis inhibitory protein
- Keyword (es)
- Anticanceroso Apoptosis Compuesto no péptido Imidazol derivado In vitro Inhibidor Mimético Relación estructura actividad Síntesis química Tiazol derivado
- Classification
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02R Antineoplastic agents / 002B02R01 General aspects
- Discipline
- Pharmacological treatments
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 16478220
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1016/j.bmcl.2004.11.010 
https://dx.doi.org/10.1016/j.bmcl.2004.11.010
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