Synthesis of a β-amino acid pharmacophore via a β-lactam intermediate
- Author
- ANGELAUD, Rémy1 ; ZHONG, Yong-Li1 ; MALIGRES, Peter1 ; LEE, Jaemoon1 ; ASKIN, David1
[1] Merck Process Research, Merck Research Laboratories, P.O. Box 2000, Rahway, New Jersey 07065, United States - Source
Journal of organic chemistry. 2005, Vol 70, Num 5, pp 1949-1952, 4 p ; ref : 24 ref
- CODEN
- JOCEAH
- ISSN
- 0022-3263
- Scientific domain
- Biochemistry, molecular biology, biophysics; Organic chemistry
- Publisher
- American Chemical Society, Washington, DC
- Publication country
- United States
- Document type
- Article
- Language
- English
- Keyword (fr)
- Aminoacide Composé chiral Hétérocycle azote Lactame Stéréosélectivité Synthèse chimique β-Lactamines Butanoïque acide(43-[t-butoxycarbonylamino]-[2,5-difluorophényl]) Pharmacophore
- Keyword (en)
- Aminoacid Chiral compound Nitrogen heterocycle Lactam Stereoselectivity Chemical synthesis β-Lactams
- Keyword (es)
- Aminoácido Compuesto quiral Heterociclo nitrógeno Lactamo Estereoselectividad Síntesis química β-Lactams
- Classification
- Pascal
- 001 Exact sciences and technology / 001C Chemistry / 001C03 Organic chemistry / 001C03C Preparations and properties / 001C03C02 Aliphatic compounds
- Discipline
- Organic chemistry
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 16578913
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1021/jo048249c 
https://dx.doi.org/10.1021/jo048249c
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