Structure-activity relationships of the oxindole growth hormone secretagogues
- Author
- TOKUNAGA, Teruhisa1 ; HUME, W. Ewan1 ; NAGAMINE, Jun1 ; KAWAMURA, Tetsuya1 ; TAIJI, Mutsuo1 ; NAGATA, Ryu1
[1] Research Division, Sumitomo Pharmaceuticals Co., Ltd, 1-98 Kasugade Naka 3-chome, Konohana-ku, Osaka 554-0022, Japan - Source
Bioorganic & medicinal chemistry letters (Print). 2005, Vol 15, Num 7, pp 1789-1792, 4 p
- ISSN
- 0960-894X
- Scientific domain
- Biochemistry, molecular biology, biophysics; Pharmacology drugs
- Publisher
- Elsevier, Oxford
- Publication country
- United Kingdom
- Document type
- Article
- Language
- English
- Keyword (fr)
- Affinité Agoniste Amine tertiaire Animal Benzène dérivé Composé aromatique Composé bicyclique Ghréline Hétérocycle azote In vitro In vivo Lactame Poids corporel Rat Relation structure activité Récepteur biologique Récepteur hormonal STH-RH Synthèse chimique Voie orale Indolin-2-one dérivé Indoline-6-carboxamide(3-[2,4-dichlorophényl]-1-[2-(diéthylamino)éthyl]-3-hydroxy-4-trifluorométhyl) chlorhydrate Chlore Composé organique Fluor Composé organique Mammalia Rodentia Vertebrata
- Keyword (en)
- Affinity Agonist Tertiary amine Animal Benzene derivatives Aromatic compound Bicyclic compound Ghrelin Nitrogen heterocycle In vitro In vivo Lactam Body weight Rat Structure activity relation Biological receptor Hormonal receptor Somatotropin releasing factor Chemical synthesis Oral administration Chlorine Organic compounds Fluorine Organic compounds Mammalia Rodentia Vertebrata
- Keyword (es)
- Afinidad Agonista Amina terciaria Animal Benceno derivado Compuesto aromático Compuesto bicíclico Grelina Heterociclo nitrógeno In vitro In vivo Lactamo Peso corporal Rata Relación estructura actividad Receptor biológico Receptor hormonal STH-RH Síntesis química Vía oral Cloro Compuesto orgánico Fluor Compuesto orgánico Mammalia Rodentia Vertebrata
- Classification
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02O Hormones. Endocrine system
- Discipline
- Pharmacological treatments
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 16626913
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1016/j.bmcl.2005.02.042 
https://dx.doi.org/10.1016/j.bmcl.2005.02.042
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