Synthesis and evaluation of potential inhibitors of eIF4E cap binding to 7-methyl GTP
- Author
- GHOSH, Phalguni1 ; PARK, Chunkyung1 ; PETERSON, Mark S2 ; BITTERMAN, Peter B2 ; POLUNOVSKY, Vitaly A2 ; WAGNER, Carston R1
[1] Department of Medicinal Chemistry, University of Minnesota, Minneapolis, MN 55455, United States
[2] Department of Medicine, University of Minnesota, Minneapolis, MN 55455, United States - Source
Bioorganic & medicinal chemistry letters (Print). 2005, Vol 15, Num 8, pp 2177-2180, 4 p
- ISSN
- 0960-894X
- Scientific domain
- Biochemistry, molecular biology, biophysics; Pharmacology drugs
- Publisher
- Elsevier, Oxford
- Publication country
- United Kingdom
- Document type
- Article
- Language
- English
- Keyword (fr)
- Activité biologique Chimiothèque Facteur initiation eIF4E GTP In vitro Inhibiteur Initiation traduction Nucléotide Phosphonate organique Phosphoramidate organique Phosphore Composé organique Purine nucléoside RNA messager Synthèse chimique α-Aminoacide Guanosine dérivé
- Keyword (en)
- Biological activity Chemical compound library Initiation factor eIF4E GTP In vitro Inhibitor Translation initiation Nucleotide Organic phosphonate Organic amidophosphate Phosphorus Organic compounds Purine nucleoside Messenger RNA Chemical synthesis α-Aminoacid
- Keyword (es)
- Actividad biológica Quimioteca Factor iniciación eIF4E GTP In vitro Inhibidor Iniciación traducción Nucleótido Fosfonato orgánico Fosforamidato orgánico Fósforo Compuesto orgánico Purina nucleósido RNA mensajero Síntesis química α-Aminoácido
- Classification
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02R Antineoplastic agents / 002B02R01 General aspects
- Discipline
- Pharmacological treatments
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 16687420
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1016/j.bmcl.2005.01.080 
https://dx.doi.org/10.1016/j.bmcl.2005.01.080
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