Synthesis and benzodiazepine receptor affinity of derivatives of the new tricyclic heteroaromatic system pyrido[3',2'5,6]thiopyrano[4,3-c]pyridazin-3(2H,5H)-one
- Author
- PRIMOFIORE, Giampaolo1 ; DA SETTIMO, Federico1 ; MARINI, Anna Maria1 ; SIMORINI, Francesca1 ; LA MOTTA, Concettina1 ; TALIANI, Sabrina1 ; LANERI, Sonia2 ; TRINCAVELLI, Letizia3 ; MARTINI, Claudia3
[1] Dipartimento di Scienze Farmaceutiche, Université di Pisa, Pisa, Italy
[2] Dipartimento di Chimica Farmaceutica e Tossicologica, Università di Napoli Federico II, Napoli, Italy
[3] Dipartimento di Psichiatria, Neurobiologia, Farmacologia e Biotecnologie, Università di Pisa, Pisa, Italy - Source
Archiv der Pharmazie (Weinheim). 2005, Vol 338, Num 2-3, pp 126-132, 7 p ; ref : 24 ref
- CODEN
- ARPMAS
- ISSN
- 0365-6233
- Scientific domain
- Organic chemistry; Pharmacology drugs
- Publisher
- Wiley-VCH, Weinheim
- Publication country
- Germany
- Document type
- Article
- Language
- English
- Author keyword
- Benzothiopyranopyridazinones Binding GABAA/Benzodiazepine receptor Pyridothiopyranopyridazinone Synthesis
- Keyword (fr)
- Activité biologique Affinité Animal Composé tricyclique Hétérocycle soufre azote In vitro Récepteur benzodiazépinique Récepteur gabaergique A Synthèse chimique Système nerveux central Benzothiopyranopyridazine Pyrido[3',2':5,6]thiopyrano[4,3-c]pyridazine dérivé Pyridothiopyranopyridazine
- Keyword (en)
- Biological activity Affinity Animal Tricyclic compound Sulfur nitrogen heterocycle In vitro Benzodiazepine receptor Gabaergic receptor A Chemical synthesis Central nervous system
- Keyword (es)
- Actividad biológica Afinidad Animal Compuesto tricíclico Heterociclo azufre nitrógeno In vitro Receptor benzodiazepínico Receptor gabaminérgico A Síntesis química Sistema nervioso central
- Classification
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02B Neuropharmacology / 002B02B09 Neurotransmitters. Neurotransmission. Receptors / 002B02B09D Gabaergic and benzodiazepinic system
- Discipline
- Pharmacological treatments
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 16737149
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1002/ardp.200400948 
https://dx.doi.org/10.1002/ardp.200400948
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