Synthesis and antibacterial activity of hydrolytically stable (-)-epicatechin gallate analogues for the modulation of β-lactam resistance in Staphylococcus aureus
- Author
- ANDERSON, James C1 ; HEADLEY, Catherine1 ; STAPLETON, Paul D2 ; TAYLOR, Peter W2
[1] School of Chemistry, University of Nottingham, Nottingham NG7 2RD, United Kingdom
[2] Microbiology Group, School of Pharmacy, University of London, 29-39 Brunswick Square, London WC1 1AX, United Kingdom - Source
Bioorganic & medicinal chemistry letters (Print). 2005, Vol 15, Num 10, pp 2633-2635, 3 p
- ISSN
- 0960-894X
- Scientific domain
- Biochemistry, molecular biology, biophysics; Pharmacology drugs
- Publisher
- Elsevier, Oxford
- Publication country
- United Kingdom
- Document type
- Article
- Language
- English
- Author keyword
- (-)-Epicatechingallate analogues MRSA β-Lactam antibiotics
- Keyword (fr)
- Acide phénolique Activité biologique Amine Antibactérien Association médicamenteuse Carboxamide Epimère Ester Gallique acide dérivé In vitro Interaction médicamenteuse Modification chimique Modulation Méticilline Oxacilline Polyphénol Résistance Staphylococcus aureus Synthèse chimique β-Lactamines Epicatéchine gallate Souche résistante méticilline Bactérie Micrococcaceae Micrococcales
- Keyword (en)
- Phenolic acid Biological activity Amine Antibacterial agent Drug combination Carboxamide Epimer Ester Gallic acid derivatives In vitro Drug interaction Chemical modification Modulation Meticillin Oxacillin Polyphenol Resistance Staphylococcus aureus Chemical synthesis β-Lactams Bacteria Micrococcaceae Micrococcales
- Keyword (es)
- Acido fenólico Actividad biológica Amina Antibacteriano Asociación medicamentosa Carboxamida Epímero Ester Gálico ácido derivado In vitro Interacción medicamentosa Modificación química Modulación Meticilina Oxacilina Polifenol Resistencia Staphylococcus aureus Síntesis química β-Lactams Bacteria Micrococcaceae Micrococcales
- Classification
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02S Antibiotics. Antiinfectious agents. Antiparasitic agents / 002B02S02 Antibacterial agents
- Discipline
- Pharmacological treatments
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 16746179
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1016/j.bmcl.2005.03.063 
https://dx.doi.org/10.1016/j.bmcl.2005.03.063
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