Synthesis and antibacterial activity of 5-methoxy- and 5-hydroxy-6-fluoro-1,8-naphthyridone-3-carboxylic acid derivatives
- Author
- HANSEN, T. Matthew1 ; GU, Yu-Gui1 ; REHM, Tamara M1 ; DANDLIKER, Peter J1 ; CHOVAN, Linda E1 ; BUI, Mai H1 ; NILIUS, Angela M1 ; BEUTEL, Bruce A1
[1] Global Pharmaceutical Research and Development, Abbott Laboratories, Abbott Park, IL 60064, United States - Source
Bioorganic & medicinal chemistry letters (Print). 2005, Vol 15, Num 11, pp 2716-2719, 4 p
- ISSN
- 0960-894X
- Scientific domain
- Biochemistry, molecular biology, biophysics; Pharmacology drugs
- Publisher
- Elsevier, Oxford
- Publication country
- United Kingdom
- Document type
- Article
- Language
- English
- Author keyword
- 1,8-Naphthyridone antibiotics Novel ribosome inhibitors
- Keyword (fr)
- Antibactérien Azétidine dérivé Composé bicyclique Haemophilus influenzae Hétérocycle azote In vitro Inhibition Naphtyridine dérivé Relation structure activité Streptococcus pneumoniae Synthèse chimique Synthèse protéique 1,8-Naphtyrid-4-one dérivé 1,8-Naphtyridine-3-carboxylique acide dérivé Bactérie Fluor Composé organique Micrococcales Pasteurellaceae Streptococcaceae
- Keyword (en)
- Antibacterial agent Azetidine derivatives Bicyclic compound Haemophilus influenzae Nitrogen heterocycle In vitro Inhibition Naphtyridine derivatives Structure activity relation Streptococcus pneumoniae Chemical synthesis Protein synthesis Bacteria Fluorine Organic compounds Micrococcales Pasteurellaceae Streptococcaceae
- Keyword (es)
- Antibacteriano Compuesto bicíclico Haemophilus influenzae Heterociclo nitrógeno In vitro Inhibición Relación estructura actividad Streptococcus pneumoniae Síntesis química Síntesis proteica Bacteria Fluor Compuesto orgánico Micrococcales Pasteurellaceae Streptococcaceae
- Classification
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02S Antibiotics. Antiinfectious agents. Antiparasitic agents / 002B02S02 Antibacterial agents
- Discipline
- Pharmacological treatments
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 16810653
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1016/j.bmcl.2005.04.007 
https://dx.doi.org/10.1016/j.bmcl.2005.04.007
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