Synthesis of an N-acyl sulfamate analog of luciferyl-AMP : A stable and potent inhibitor of firefly luciferase
- Author
- BRANCHINI, Bruce R1 ; MURTIASHAW, Martha H1 ; CARMODY, Jill N1 ; MYGATT, Emily E1 ; SOUTHWORTH, Tara L1
[1] Department of Chemistry, Connecticut College, 270 Mohegun Avenue, New London, CT06320, United States - Source
Bioorganic & medicinal chemistry letters (Print). 2005, Vol 15, Num 17, pp 3860-3864, 5 p ; ref : 29 ref
- ISSN
- 0960-894X
- Scientific domain
- Biochemistry, molecular biology, biophysics; Pharmacology drugs
- Publisher
- Elsevier, Oxford
- Publication country
- United Kingdom
- Document type
- Article
- Language
- English
- Author keyword
- Acyl-adenylate Adenylate-forming Bioluminescence Chymotrypsin Firefly Inhibitor Limited proteolysis Luciferase Sulfamate Sulfonamide
- Keyword (fr)
- Activité biologique Amidosulfate organique Benzothiazole dérivé Bioluminescence Changement conformation Chymotrypsin Conformation In vitro Inhibiteur enzyme Photinus-luciferin 4-monooxygenase (ATP-hydrolysing) Protéine Purine nucléoside Réaction catalytique Synthèse chimique Thiazole dérivé Adénosine 5p-amidosulfate[2-(6-hydroxybenzothiazol-3-yl)thiazole-4-carbonyl] Adénosine dérivé Enzyme Hydrolases Oxidoreductases Peptidases Serine endopeptidases
- Keyword (en)
- Biological activity Organic amidosulfate Benzothiazole derivatives Bioluminescence Conformational changes Chymotrypsin Conformation In vitro Enzyme inhibitor Photinus-luciferin 4-monooxygenase (ATP-hydrolysing) Protein Purine nucleoside Catalytic reaction Chemical synthesis Thiazole derivatives Enzyme Hydrolases Oxidoreductases Peptidases Serine endopeptidases
- Keyword (es)
- Actividad biológica Amidosulfato orgánico Benzotiazol derivado Bioluminiscencia Chymotrypsin Conformación In vitro Inhibidor enzima Photinus-luciferin 4-monooxygenase (ATP-hydrolysing) Proteína Purina nucleósido Reacción catalítica Síntesis química Tiazol derivado Enzima Hydrolases Oxidoreductases Peptidases Serine endopeptidases
- Classification
- Pascal
- 002 Biological and medical sciences / 002A Fundamental and applied biological sciences. Psychology / 002A02 Analytical, structural and metabolic biochemistry / 002A02E Enzymes and enzyme inhibitors / 002A02E02 Oxidoreductases
- Discipline
- Analytical, structural and metabolic biochemistry
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 16984216
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1016/j.bmcl.2005.05.115 
https://dx.doi.org/10.1016/j.bmcl.2005.05.115
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