Synthesis of tripeptides as potent Yersinia protein tyrosine phosphatase inhibitors
- Author
- LEE, Kyeong1 2 ; BOOVANAHALLI, Shanthaveerappa K2 ; JUNG JUN LEE2 ; BURKE, Terrence R1 ; NAM, Ky-Youb3 ; KANG, Sang-Uk1 ; LEE, Mijeoung2 ; PHAN, Jason4 ; LI WU5 ; WAUGH, David S4 ; ZHANG, Zhong-Yin5 ; KYOUNG TAI NO3
[1] Laboratory of Medicinal Chemistry, NCI, NIH, NCI-Frederick, Frederick, MD 21702, United States
[2] Laboratory of Anticancer Research, KRIBB, Duejeon 305-333, Korea, Republic of
[3] Department of Biotechnology, Yonsei University, Seodaemun-gu, Seoul 120-749, Korea, Republic of
[4] Macromolecular Crystallography Laboratory, NCI, NIH, NCI-Frederick, Frederick, MD 21702, United States
[5] Department of Molecular Pharmacology, Albert Einstein Medical School, Bronx, NY 10461, United States - Source
Bioorganic & medicinal chemistry letters (Print). 2005, Vol 15, Num 18, pp 4037-4042, 6 p
- ISSN
- 0960-894X
- Scientific domain
- Biochemistry, molecular biology, biophysics; Pharmacology drugs
- Publisher
- Elsevier, Oxford
- Publication country
- United Kingdom
- Document type
- Article
- Language
- English
- Author keyword
- Bioterrorism PTPIB Tripeptides YopH pTyr mimetics
- Keyword (fr)
- Activité biologique Bioterrorisme Carboxamide Complexe enzyme inhibiteur Homme Indole dérivé Inhibiteur enzyme Mimétique Mode liaison Modèle moléculaire Modélisation Peptide Protein-tyrosine-phosphatase Pseudopeptide Synthèse chimique Transduction signal Tripeptide Yersinia Isoglutamine dérivé Leucine dérivé Phosphotyrosine Tyrosine dérivé Bactérie Enterobacteriaceae Enzyme Esterases Hydrolases Phosphoric monoester hydrolases
- Keyword (en)
- Biological activity Bioterrorism Carboxamide Inhibitor enzyme complex Human Indole derivatives Enzyme inhibitor Mimetic Binding mode Molecular model Modeling Peptides Protein-tyrosine-phosphatase Pseudopeptide Chemical synthesis Signal transduction Tripeptide Yersinia Bacteria Enterobacteriaceae Enzyme Esterases Hydrolases Phosphoric monoester hydrolases
- Keyword (es)
- Actividad biológica Bioterrorismo Carboxamida Complejo enzima inhibidor Hombre Indol derivado Inhibidor enzima Mimético Modo de enlace Modelo molecular Modelización Péptido Protein-tyrosine-phosphatase Seudopéptido Síntesis química Transducción señal Tripéptido Yersinia Bacteria Enterobacteriaceae Enzima Esterases Hydrolases Phosphoric monoester hydrolases
- Classification
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02S Antibiotics. Antiinfectious agents. Antiparasitic agents / 002B02S02 Antibacterial agents
- Discipline
- Pharmacological treatments
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 17018573
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1016/j.bmcl.2005.06.027 
https://dx.doi.org/10.1016/j.bmcl.2005.06.027
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