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Analysis of structure-activity relationships for the 'B-region' of N-(4-t-butylbenzyl)-N'-[4-(methylsulfonylamino)benzyl ]- thiourea analogues as TRPV1 antagonists

Author
LEE, Jeewoo1 ; JIN, Mi-Kyoung1 ; KIM, Sung-Eun1 ; SUH, Young-Ger1 ; LEE, Yong-Sil1 ; KIM, Young-Ho2 ; HA, Hee-Jin2 ; TOTH, Attila3 ; PEARCE, Larry V3 ; TRAN, Richard3 ; SZABO, Tamas3 ; WELTER, Jacqueline D3 ; KANG, Sang-Uk1 ; LUNDBERG, Daniel J3 ; YUN WANG3 ; LAZAR, Jozsef3 ; PAVLYUKOVETS, Vladimir A3 ; MORGAN, Matthew A3 ; BLUMBERG, Peter M3 ; SU YEON KIM1 ; LEE, Jiyoun1 ; SHIN, Myoungyoup1 ; HWANG, Jaemin1 ; CHO, Sookhyun1 ; CHOI, Yeon-Sil1 ; CHOI, Hyun-Kyung1
[1] Research Institute of Pharmaceutical Sciences, College of Pharmacy, Seoul National University, Seoul 151-742, Korea, Republic of
[2] Digitalbiotech, Ansan, Kyounggi-Do 425-839, Korea, Republic of
[3] Laboratory of Cellular Carcinogenesis and Tumor Promotion, Center for Cancer Research, National Cancer Institute, NIH, Bethesda, MD 20892, United States
Source

Bioorganic & medicinal chemistry letters (Print). 2005, Vol 15, Num 18, pp 4143-4150, 8 p

ISSN
0960-894X
Scientific domain
Biochemistry, molecular biology, biophysics; Pharmacology drugs
Publisher
Elsevier, Oxford
Publication country
United Kingdom
Document type
Article
Language
English
Author keyword
Capsaicin Molecular modeling Resiniferatoxin TRPV1 antagonist Vanilloid Receptor 1 antagonist
Keyword (fr)
Antagoniste Benzène dérivé Capsaïcine In vitro Modèle moléculaire Modélisation Prédiction Relation structure activité Récepteur vanilloïde VR1 Thiourées Récepteur vanilloïde TRPV1 Résinifératoxine Thiourée(1-[4-t-butylbenzyl]-3-[4-(mésylamino)benzyl])
Keyword (en)
Antagonist Benzene derivatives Capsaicin In vitro Molecular model Modeling Prediction Structure activity relation VR1 vanilloid receptor Thioureas TRPV1 vanilloid receptor
Keyword (es)
Antagonista Benceno derivado Capsicina In vitro Modelo molecular Modelización Predicción Relación estructura actividad Receptor vaniloide VR1 Tioureas
Classification
Pascal
002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02B Neuropharmacology / 002B02B09 Neurotransmitters. Neurotransmission. Receptors / 002B02B09G Miscellaneous

Discipline
Pharmacological treatments
Origin
Inist-CNRS
Database
PASCAL
INIST identifier
17018593

Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS

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