Microwave-assisted synthesis of antimicrobial dihydropyridines and tetrahydropyrimidin-2-ones : Novel compounds against aspergillosis
- Author
- CHHILLAR, Anil K1 ; ARYA, Pragya2 ; WATTERSON, Arthur C4 ; PARMAR, Virinder S2 4 ; PRASAD, Ashok K2 ; SHARMA, Gainda L1 ; MUKHERJEE, Chandrani2 ; KUMAR, Pankaj2 3 ; YADAV, Yogesh2 3 ; SHARMA, Ajendra K2 4 ; YADAV, Vibha1 ; GUPTA, Jyotsana1 ; DABUR, Rajesh1 ; JHA, Hirday N3
[1] Institute of Genomics & Integrative Biology, Mall Road, Delhi 110 007, India
[2] Bioorganic Laboratory, Department of Chemistry, University of Delhi, Delhi 110 007, India
[3] Department of Chemistry, MMH College, CCS University, Meerut 250 002, India
[4] Institute for Nano Science and Engineering Technology, Department of Chemistry, University of Massachusetts, Lowell, MA 01854, United States - Source
Bioorganic & medicinal chemistry. 2006, Vol 14, Num 4, pp 973-981, 9 p ; ref : 45 ref
- ISSN
- 0968-0896
- Scientific domain
- Biochemistry, molecular biology, biophysics; Pharmacology drugs
- Publisher
- Elsevier Science, Oxford
- Publication country
- United Kingdom
- Document type
- Article
- Language
- English
- Author keyword
- 4-Aryl-1,2,3,4-tetrahydropyrimidinone 4-Aryl-1,4-dihydropyridine Antifungal agent Aspergillosis Microwave-assisted reaction
- Keyword (fr)
- Activité biologique Amphotéricine B Antifongique Antimicrobien Aspergillus fumigatus Candida albicans Chauffage hyperfréquence Cytotoxicité Dihydropyridine dérivé Erythrocyte Homme Hémolyse In vitro Pyrimidine dérivé Pyrimidinone dérivé Relation structure activité Synthèse chimique Toxicité Pyridine-3,5-dicarboxylique acide(1,4-dihydro-2,6-diméthyl-4-[4-méthoxyphényl]) ester diéthyle Pyrimidine-5-carboxylique acide dérivé Fungi Imperfecti Fungi Thallophyta
- Keyword (en)
- Biological activity Amphotericin B Antifungal agent Antimicrobial agent Aspergillus fumigatus Candida albicans Microwave heating Cytotoxicity Dihydropyridine derivatives Red blood cell Human Hemolysis In vitro Pyrimidine derivatives Pyrimidone derivatives Structure activity relation Chemical synthesis Toxicity Fungi Imperfecti Fungi Thallophyta
- Keyword (es)
- Actividad biológica Amfotericina B Antifúngico Antimicrobiano Aspergillus fumigatus Candida albicans Calentamiento hiperfrecuencia Citotoxicidad Dihidropiridine derivado Eritrocito Hombre Hemólisis In vitro Pirimidina derivado Relación estructura actividad Síntesis química Toxicidad Fungi Imperfecti Fungi Thallophyta
- Classification
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02S Antibiotics. Antiinfectious agents. Antiparasitic agents / 002B02S01 General aspects
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02S Antibiotics. Antiinfectious agents. Antiparasitic agents / 002B02S04 Antifungal agents
- Discipline
- Pharmacological treatments
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 17554784
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1016/j.bmc.2005.09.014 
https://dx.doi.org/10.1016/j.bmc.2005.09.014
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