Arylpiperazines with N-acylated amino acids as 5-HT1A receptor ligands
- Author
- ZAJDEL, Pawel1 2 ; SUBRA, Gilles1 ; BOJARSKI, Andrzej J3 ; DUSZYNSKA, Beata3 ; PAWLOWSKI, Maciej2 ; MARTINEZ, Jean1
[1] Laboratoire des Aminoacides, Peptides et Protéines (LAPP), UMR 5810, Faculté de Pharmacie, Université Montpellier I et II, 15 Avenue Charles Flahault, 34060 Montpellier, France
[2] Department of Medicinal Chemistry, Jagiellonian University Medical Collège, 9 Medyczna Street, 30-688 Kraków, Poland
[3] Department of Medicinal Chemistry, Institute of Phcirinacology, Poiish Aia of Sciences, 12 Sinelmi Street, 31-343 Krakôw, Poland - Source
Bioorganic & medicinal chemistry letters (Print). 2006, Vol 16, Num 13, pp 3406-3410, 5 p
- ISSN
- 0960-894X
- Scientific domain
- Biochemistry, molecular biology, biophysics; Pharmacology drugs
- Publisher
- Elsevier, Oxford
- Publication country
- United Kingdom
- Document type
- Article
- Language
- English
- Author keyword
- 5-HT1A receptor ligands BAL linker Fujila- Ban analysis Long-chain arylpiperazines Pyroglutamates Solid-phase synthesis Succinimides
- Keyword (fr)
- Acylation Aminoacide Chaîne longue Chimiothèque Criblage Imide In vitro In vivo Ligand Phase solide Pipérazine dérivé Relation structure activité Récepteur sérotoninergique 5-HT1A Synthèse chimique Asparaginamide dérivé Asparagine dérivé Bras espaceur Proline dérivé Pyroglutamique acide dérivé Succinimide dérivé
- Keyword (en)
- Acylation Aminoacid Long chain Chemical compound library Screening Imide In vitro In vivo Ligand Solid phase Piperazine derivatives Structure activity relation 5-HT1A Serotonine receptor Chemical synthesis Spacer arm
- Keyword (es)
- Acilación Aminoácido Cadena larga Quimioteca Cernido Imida In vitro In vivo Ligando Fase sólida Piperazina derivado Relación estructura actividad Receptor serotoninérgico 5-HT1A Síntesis química
- Classification
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02B Neuropharmacology / 002B02B09 Neurotransmitters. Neurotransmission. Receptors / 002B02B09C Serotoninergic system
- Discipline
- Pharmacological treatments
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 17800214
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1016/j.bmcl.2006.04.035 
https://dx.doi.org/10.1016/j.bmcl.2006.04.035
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