Redefining the structure-activity relationships of 2,6-methano-3-benzazocines. 4. Opioid receptor binding properties of 8-[N-(4'-phenyl)-phenethylcarboxamido] analogues of cyclazocine and ethylketocycalzocine
- Author
- WENTLAND, Mark P1 ; VANALSTINE, Melissa1 ; KUCEJKO, Robert1 ; RONGLIANG LOU1 ; COHEN, Dana J2 ; PARKHILL, Amy L2 ; BIDLACK, Jean M2
[1] Department of Chemistry and Chemical Biology, Rensselaer Polytechnic Institute, Troy, New York 12180, United States
[2] Department of Pharmacology and Physiology, School of Medicine and Dentistry, University of Rochester, Rochester, New York 14642, United States - Source
Journal of medicinal chemistry (Print). 2006, Vol 49, Num 18, pp 5635-5639, 5 p ; ref : 9 ref
- CODEN
- JMCMAR
- ISSN
- 0022-2623
- Scientific domain
- Pharmacology drugs
- Publisher
- American Chemical Society, Washington, DC
- Publication country
- United States
- Document type
- Article
- Language
- English
- Keyword (fr)
- Benzomorphane dérivé Biphényle dérivé Carboxamide Cyclazocine Cyclopropane dérivé Enantiomère Fixation biologique In vitro Interaction moléculaire Relation structure activité Récepteur opiacé Synthèse chimique 2,6-Méthano-3-benzoazocine dérivé 2,6-Méthano-3-benzoazocine-8-carboxamide dérivé
- Keyword (en)
- Benzomorphane derivatives Biphenyl derivatives Carboxamide Cyclazocine Cyclopropane derivatives Enantiomer Biological fixation In vitro Molecular interaction Structure activity relation Opioid receptor Chemical synthesis
- Keyword (es)
- Benzomorfano derivado Bifenilo derivado Carboxamida Ciclazocina Ciclopropano derivado Enantiómero Fijación biológica In vitro Interacción molecular Relación estructura actividad Receptor opiáceo Síntesis química
- Classification
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02B Neuropharmacology / 002B02B09 Neurotransmitters. Neurotransmission. Receptors / 002B02B09F Peptidergic system (neuropeptide, opioid peptide, opiates...). Adenosinergic and purinergic systems
- Discipline
- Pharmacological treatments
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 18073850
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1021/jm060278n 
https://dx.doi.org/10.1021/jm060278n
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