Inhibition of Src kinase activity by 7-ethynyl-4-phenylamino-3-quinolinecarbonitriles : Identification of SKS-927
- Author
- BOSCHELLI, Diane H1 ; BARRIOS SOSA, Ana Carolina1 ; GOLAS, Jennifer M2 ; BOSCHELLI, Frank2
[1] Wyeth Research, Chemical and Screening Sciences, 401 N. Middletown Road, Pearl River, NY 10965, United States
[2] Wyeth Research, Oncology, 401 N. Middletown Road, Pearl River, NY 10965, United States - Source
Bioorganic & medicinal chemistry letters (Print). 2007, Vol 17, Num 5, pp 1358-1361, 4 p
- ISSN
- 0960-894X
- Scientific domain
- Biochemistry, molecular biology, biophysics; Pharmacology drugs
- Publisher
- Elsevier, Oxford
- Publication country
- United Kingdom
- Document type
- Article
- Language
- English
- Author keyword
- 3-Quinolinecarbonitrile Src
- Keyword (fr)
- Activité biologique Amine aromatique Aniline dérivé Anticancéreux Chlore composé organique Composé acétylénique Inhibition Nitrile Pipérazine dérivé Protein-tyrosine kinase Quinoléine dérivé Synthèse chimique Transduction signal Quinoléine-3-carbonitrile dérivé Enzyme Transferases
- Keyword (en)
- Biological activity Aromatic amine Aniline derivatives Antineoplastic agent Organic chlorine compounds Acetylenic compound Inhibition Nitrile Piperazine derivatives Protein-tyrosine kinase Quinoline derivatives Chemical synthesis Signal transduction Enzyme Transferases
- Keyword (es)
- Actividad biológica Amina aromática Anilina derivado Anticanceroso Compuesto acetilénico Inhibición Nitrilo Piperazina derivado Protein-tyrosine kinase Quinolina derivado Síntesis química Transducción señal Enzima Transferases
- Classification
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02R Antineoplastic agents / 002B02R01 General aspects
- Discipline
- Pharmacological treatments
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 18573758
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1016/j.bmcl.2006.11.077 
https://dx.doi.org/10.1016/j.bmcl.2006.11.077
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