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Comparative evaluation of central Muscarinic receptor binding activity by oxybutynin, tolterodine and darifenacin used to treat overactive bladder

Author
OKI, Tomomi1 ; KAGEYAMA, Aiko1 ; TAKAGI, Yukiko1 ; UCHIDA, Shinya1 ; YAMADA, Shizuo1
[1] Department of Pharmacokinetics and Pharmacodynamics and Center of Excellence Program in the 21st Centry, School of Pharmaceutical Sciences, University of Shizuoka, Suruga-ku, Shizuoka, Japan
Source

The Journal of urology. 2007, Vol 177, Num 2, pp 766-770, 5 p ; ref : 20 ref

CODEN
JOURAA
ISSN
0022-5347
Scientific domain
Urology, nephrology
Publisher
Lippincott Williams & Wilkins, Hagerstown, MD
Publication country
United States
Document type
Article
Language
English
Author keyword
bladder; mice; receptors muscarinic; cholinergic antagonists; cerebral cortex
Keyword (fr)
Activité biologique Animal Antagoniste Cortex cérébral Darifénacine Etude comparative Evaluation Liaison Oxybutynine Récepteur biologique Récepteur muscarinique Souris Spasmolytique Toltérodine Traitement Urologie Vessie hyperactive Vessie urinaire Néphrologie Appareil urinaire pathologie Appareil urinaire Encéphale Mammalia Parasympatholytique Rodentia Récepteur cholinergique Récepteur muscarinique M3 Système nerveux central Vertebrata Vessie pathologie Voie urinaire pathologie
Keyword (en)
Biological activity Animal Antagonist Cerebral cortex Darifenacin Comparative study Evaluation Binding Oxybutynin Biological receptor Muscarinic receptor Mouse Antispasmodic agent Tolterodine Treatment Urology Overactive bladder Urinary bladder Nephrology Urinary system disease Urinary system Encephalon Mammalia Parasympatholytic Rodentia Cholinergic receptor M3 Muscarinic receptor Central nervous system Vertebrata Bladder disease Urinary tract disease
Keyword (es)
Actividad biológica Animal Antagonista Corteza cerebral Darifenacina Estudio comparativo Evaluación Enlace Oxibutinina Receptor biológico Receptor muscarínico Ratón Espasmolítico Tolterodina Tratamiento Urología Vejiga hiperactiva Vejiga Nefrología Aparato urinario patología Aparato urinario Encéfalo Mammalia Parasimpatolítico Rodentia Receptor colinérgico Receptor muscarínico M3 Sistema nervioso central Vertebrata Vejiga patología Vía urinaria patología
Classification
Pascal
002 Biological and medical sciences / 002B Medical sciences / 002B14 Nephrology. Urinary tract diseases / 002B14E Urinary system involvement in other diseases. Miscellaneous / 002B14E02 Urinary tract. Prostate gland

Discipline
Nephrology. Urinary tract diseases
Origin
Inist-CNRS
Database
PASCAL
INIST identifier
18825671

Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS

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