Regioselective synthesis of 4-and 7-alkoxyindoles from 2,3-dihalophenols : Application to the preparation of indole inhibitors of phospholipase A2
- Author
- SANZ, Roberto1 ; CASTROVIEJO, M. Pilar1 ; GUILARTE, Veronica1 ; PEREZ, Antonio1 ; FANANAS, Francisco J2
[1] Departamento de Química, Área de Química Orgánica, Facultad de Ciencias, Universidad de Burgos, Pza. Misael Bahuelos s/n, 09001-Burgos, Spain
[2] Instituto Universitario de Química Organometàlica Enrique Moles, Universidad de Oviedo, C/ Julián Clavería, 8, 33006-Oviedo, Spain - Source
Journal of organic chemistry. 2007, Vol 72, Num 14, pp 5113-5118, 6 p
- CODEN
- JOCEAH
- ISSN
- 0022-3263
- Scientific domain
- Biochemistry, molecular biology, biophysics; Organic chemistry
- Publisher
- American Chemical Society, Washington, DC
- Publication country
- United States
- Document type
- Article
- Language
- English
- Keyword (fr)
- Acétique acide dérivé Amination Amine Anisole Composé benzylique Cyclisation Halogénophénols Hétérocycle azote Indole dérivé Inhibiteur enzyme Métallation Palladium complexe Phospholipase A2 Phénols Réaction catalytique Réaction tandem Régiosélectivité Synthèse chimique Copulation Sonogashira Carboxylic ester hydrolases Enzyme Esterases Hydrolases Métal transition complexe Platinoïde Complexe
- Keyword (en)
- Acetic acid derivative Amination Amine Benzylic compound Cyclization Halophenols Nitrogen heterocycle Indole derivatives Enzyme inhibitor Metalation Palladium complex Phospholipase A2 Phenols Catalytic reaction Tandem reaction Regioselectivity Chemical synthesis Carboxylic ester hydrolases Enzyme Esterases Hydrolases Transition element complexes Platinoid Complexes
- Keyword (es)
- Acético ácido derivado Aminación Amina Compuesto benzílico Ciclización Halofenoles Heterociclo nitrógeno Indol derivado Inhibidor enzima Metalación Paladio complejo Phospholipase A2 Fenoles Reacción catalítica Reacción tándem Regioselectividad Síntesis química Carboxylic ester hydrolases Enzima Esterases Hydrolases Platinoide Complejo
- Classification
- Pascal
- 001 Exact sciences and technology / 001C Chemistry / 001C03 Organic chemistry / 001C03C Preparations and properties / 001C03C06 Heterocyclic compounds / 001C03C06B Heterocyclic compounds with only one n hetero atom and condensed derivatives
- Discipline
- Organic chemistry
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 18915963
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1021/jo070643y 
https://dx.doi.org/10.1021/jo070643y
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