A novel ketolide class : Synthesis and antibacterial activity of a lead compound
- Author
- ANDREOTTI, Daniele1 ; BIENTINESI, Ilaria1 ; BIONDI, Stefano2 ; DONATI, Daniele1 ; ERBETTI, Isabelle1 ; LOCIURO, Sergio3 ; MARCHIORO, Carla1 ; POZZAN, Alfonso1 ; RATTI, Emiliangelo1 ; TERRENI, Silvia1
[1] GlaxosmithKline, Medicine Research Centre, Via A Fleming 4, 37135 Verona, Italy
[2] NicOx Research Institute, Via Ariosto 21, Bresso MI 20 09, Italy
[3] Arpida Ltd. Research & Development of Anti-Infectives, Dammstrase 36, 4142 Münchenstein, Switzerland - Source
Bioorganic & medicinal chemistry letters (Print). 2007, Vol 17, Num 18, pp 5265-5269, 5 p ; ref : 30 ref
- ISSN
- 0960-894X
- Scientific domain
- Biochemistry, molecular biology, biophysics; Pharmacology drugs
- Publisher
- Elsevier, Oxford
- Publication country
- United Kingdom
- Document type
- Article
- Language
- English
- Author keyword
- Antibacterial GW680788X Ketolides Macrolides
- Keyword (fr)
- Activité biologique Antibactérien Antibiotique Clarithromycine Composé bicyclique Etude comparative Hétérocycle oxygène In vitro Kétolide Macrolide Synthèse chimique
- Keyword (en)
- Biological activity Antibacterial agent Antibiotic Clarithromycin Bicyclic compound Comparative study Oxygen heterocycle In vitro Ketolide Macrolide Chemical synthesis
- Keyword (es)
- Actividad biológica Antibacteriano Antibiótico Claritromicina Compuesto bicíclico Estudio comparativo Heterociclo oxígeno In vitro Ketolide Macrólido Síntesis química
- Classification
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02S Antibiotics. Antiinfectious agents. Antiparasitic agents / 002B02S02 Antibacterial agents
- Discipline
- Pharmacological treatments
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 19021301
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1016/j.bmcl.2007.02.019 
https://dx.doi.org/10.1016/j.bmcl.2007.02.019
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