A refined agonist pharmacophore for protease activated receptor 2
- Author
- BARRY, Grant D1 ; SUEN, Jacky Y1 ; LOW, Heng Boon1 ; PFEIFFER, Bernhard1 ; FLANAGAN, Bernadine1 ; HALILI, Maria1 ; LE, Giang T1 ; FAIRLIE, David P1
[1] Centre for Drug Design and Development, Institute for Molecular Bioscience, University of Queensland, Brisbane, Qld. 4072, Australia - Source
Bioorganic & medicinal chemistry letters (Print). 2007, Vol 17, Num 20, pp 5552-5557, 6 p
- ISSN
- 0960-894X
- Scientific domain
- Biochemistry, molecular biology, biophysics; Pharmacology drugs
- Publisher
- Elsevier, Oxford
- Publication country
- United Kingdom
- Document type
- Article
- Language
- English
- Author keyword
- Agonist Fluorescence Inflammation PAR1 PAR2
- Keyword (fr)
- Affinité Agoniste Cellule tumorale Côlon Homme In vitro Inflammation Lignée cellulaire Modélisation Oligopeptide Peptide Relation structure activité Récepteur PAR2 Lignée HT29
- Keyword (en)
- Affinity Agonist Tumor cell Colon Human In vitro Inflammation Cell line Modeling Oligopeptides Peptides Structure activity relation PAR2 protease-activated receptor
- Keyword (es)
- Afinidad Agonista Célula tumoral Colón Hombre In vitro Inflamación Línea celular Modelización Oligopéptido Péptido Relación estructura actividad Receptor PAR2
- Classification
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02W Miscellaneous
- Discipline
- General pharmacology
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 19109515
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1016/j.bmcl.2007.08.026 
https://dx.doi.org/10.1016/j.bmcl.2007.08.026
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