Synthesis and biological activity of 1,2,4-oxadiazole derivatives : highly potent and efficacious agonists for cortical muscarinic receptors
- Author
- STREET, L. J; BAKER, R; HARLEY, E. A; BOOK, T; KNEEN, C. O; MACLEOD, A. M; MERCHANT, K. J; SHOWELL, G. A; SAUNDERS, J; HERBERT, R. H; FREEDMAN, S. B
Merck Sharp and Dohne Research Laboratories, chemistry dep., Essex CM20 2QR, United Kingdom - Source
Journal of medicinal chemistry (Print). 1990, Vol 33, Num 10, pp 2690-2697, 8 p ; ref : 31 ref
- CODEN
- JMCMAR
- ISSN
- 0022-2623
- Scientific domain
- Pharmacology drugs
- Publisher
- American Chemical Society, Washington, DC
- Publication country
- United States
- Document type
- Article
- Language
- English
- Keyword (fr)
- Activité biologique Composé bicyclique Hétérocycle azote angulaire Hétérocycle oxygène azote Parasympathomimétique 1,2,4-Oxadiazole dérivé Arecoline dérivé Azabicycloheptane dérivé
- Keyword (en)
- Biological activity Bicyclic compound Angular nitrogen heterocycle Oxygen nitrogen heterocycle Parasympathomimetic
- Keyword (es)
- Actividad biológica Compuesto bicíclico Heterociclo nitrógeno angular Heterociclo oxígeno nitrógeno Parasimpatomimético
- Classification
- Pascal
- 001 Exact sciences and technology / 001C Chemistry / 001C03 Organic chemistry / 001C03C Preparations and properties / 001C03C06 Heterocyclic compounds / 001C03C06D Heterocyclic compounds with n hetero atom and also o and/or s, se, te hetero atoms
- Discipline
- Organic chemistry
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 19539235
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1021/jm00172a003 
https://dx.doi.org/10.1021/jm00172a003
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