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A potent nonpeptide antagonist of the substance P (NK1) receptor

Author
SNIDER, R. M; CONSTANTINE, J. W; HESS, H.-J; LOWE, J. A; LONGO, K. P; LEBEL, W. S; WOODY, H. A; DROZDA, S. E; DESAI, M. C; VINICK, F. J; SPENCER, R. W
Pfizer Inc., dep. exploratory medicinal chemistry, cent. res. div., Groton CT 06340, United States
Source

Science (Washington, D.C.). 1991, Vol 251, Num 4992, pp 435-437, 3 p ; ref : 20 ref

CODEN
SCIEAS
ISSN
0036-8075
Scientific domain
Multidisciplinary
Publisher
American Association for the Advancement of Science, Washington, DC
Publication country
United States
Document type
Article
Language
English
Keyword (fr)
Antagoniste Chien Fixation ligand Hormone peptide Inhibition Marquage radioisotopique Neuropeptide Rat Relation dose réponse Récepteur hormonal Spécificité Substance P CP96,345 Récepteur NK-1 Carnivora Fissipedia Mammalia Rodentia Vertebrata
Keyword (en)
Antagonist Dog Ligand binding Peptide hormone Inhibition Radiolabelling Neuropeptide Rat Dose activity relation Hormonal receptor Specificity Substance P Carnivora Fissipedia Mammalia Rodentia Vertebrata
Keyword (es)
Antagonista Perro Fijación ligando Hormona péptido Inhibición Marcación radioisotópica Neuropéptido Rata Relación dosis respuesta Receptor hormonal Especificidad Substancia P Carnivora Fissipedia Mammalia Rodentia Vertebrata
Classification
Pascal
002 Biological and medical sciences / 002A Fundamental and applied biological sciences. Psychology / 002A04 Molecular and cellular biology / 002A04F Cell structures and functions / 002A04F03 Cell receptors / 002A04F03D Neuropeptide receptors

Discipline
Molecular and cell biology
Origin
Inist-CNRS
Database
PASCAL
INIST identifier
19640237

Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS

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