Synthesis, SAR, and antibacterial activity of novel oxazolidinone analogues possessing urea functionality
- Author
- SELVAKUMAR, N1 ; GOVINDA RAJULU, G1 ; AMARNATH, P. V. S1 ; KANDEPU, Sreenivas1 ; IQBAL, Javed1 ; CHANDRA SHEKAR REDDY, K1 ; CHANDRA CHARY, B1 ; KALYAN KUMAR, P1 ; MADHAVI, T1 ; PRAVEENA, K1 ; HARI PRASADA REDDY, K1 ; TAKHI, Mohammed1 ; MALLICK, Arundhuti1
[1] Anti-infectives Discovery Group, Discovery Research, Dr. Reddy's Laboratories Ltd, Miyapur , Hyderabad 500 049, India - Source
Bioorganic & medicinal chemistry letters (Print). 2008, Vol 18, Num 2, pp 856-860, 5 p ; ref : 11 ref
- ISSN
- 0960-894X
- Scientific domain
- Biochemistry, molecular biology, biophysics; Pharmacology drugs
- Publisher
- Elsevier, Oxford
- Publication country
- United Kingdom
- Document type
- Article
- Language
- English
- Author keyword
- Antibacterial Linezolid Oxazolidinones Urea
- Keyword (fr)
- Antibactérien Carbamate organique Cycle 5 chaînons Cycle 6 chaînons Dérivé de l'oxazolidinone Dérivé du benzène Hétérocycle azote Hétérocycle oxygène azote In vitro Relation structure activité Synthèse chimique Urées Acétamide dérivé Oxazolidin-2-one dérivé Pipérazine-1-carboxamide dérivé Dérivé de l'oxazole Fluor Composé organique
- Keyword (en)
- Antibacterial agent Organic carbamate Five membered ring Six membered ring Oxazolidinone derivative Benzene derivatives Nitrogen heterocycle Oxygen nitrogen heterocycle In vitro Structure activity relation Chemical synthesis Ureas Oxazole derivatives Fluorine Organic compounds
- Keyword (es)
- Antibacteriano Carbamato orgánico Ciclo 5 eslabones Ciclo 6 eslabones Oxazolidinona derivado Benceno derivado Heterociclo nitrógeno Heterociclo oxígeno nitrógeno In vitro Relación estructura actividad Síntesis química Ureas Oxazol derivado Fluor Compuesto orgánico
- Classification
- Pascal
- 002 Biological and medical sciences / 002B Medical sciences / 002B02 Pharmacology. Drug treatments / 002B02S Antibiotics. Antiinfectious agents. Antiparasitic agents / 002B02S02 Antibacterial agents
- Discipline
- Pharmacological treatments
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 20040276
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1016/j.bmcl.2007.09.024 
https://dx.doi.org/10.1016/j.bmcl.2007.09.024
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