Stereochemical studies on the novel monoamine oxidase B substrates (1R,6S)-and (15,6R)-3-methyl-6-phenyl-3-aza-bicycle[4,1.0]heptane
- Author
- BISSEL, Philippe1 ; KHALIL, Ashraf1 ; RIMOLD, John M2 ; IGARASHI, Kazuo1 ; EDMONDSON, Dale3 ; MILLER, Anthony1 ; CASTAGNOLI, Neal1 4
[1] Department of Chemistry, Virginia Polytechnic Institute and State University, West Campus Dr, Blacksburg, VA 24061-0212, United States
[2] Department of Medicinal Chemistry and Laboratory for Applied Drug Design and Synthesis, The University of Mississippi, MS 38677, United States
[3] The Departments of Biochemistry and Chemistry, Emory University, Atlanta, GA 30322, United States
[4] The Edward Via Collage of Osteopathic Medicine, Blacksburg, VA 24061, United States - Source
Bioorganic & medicinal chemistry. 2008, Vol 16, Num 7, pp 3557-3564, 8 p ; ref : 48 ref
- ISSN
- 0968-0896
- Scientific domain
- Biochemistry, molecular biology, biophysics; Pharmacology drugs
- Publisher
- Elsevier Science, Oxford
- Publication country
- United Kingdom
- Document type
- Article
- Language
- English
- Author keyword
- Cyclopropyl analog of MPTP Diastereoselectivity E- nantioselectivity Monoamine oxidase B
- Keyword (fr)
- Amine oxidase (flavin-containing) Composé bicyclique Diastéréosélectivité Stéréosélectivité Substrat 3-Azabicyclo[4.1.0]heptane dérivé 3-Azabicyclo[4.1.0]heptane(3-méthyl-6-phényl) Enzyme Oxidoreductases
- Keyword (en)
- Amine oxidase (flavin-containing) Bicyclic compound Diastereoselectivity Stereoselectivity Substrate Enzyme Oxidoreductases
- Keyword (es)
- Amine oxidase (flavin-containing) Compuesto bicíclico Diastereoselectividad Estereoselectividad Substrato Enzima Oxidoreductases
- Classification
- Pascal
- 002 Biological and medical sciences / 002A Fundamental and applied biological sciences. Psychology / 002A02 Analytical, structural and metabolic biochemistry / 002A02E Enzymes and enzyme inhibitors / 002A02E02 Oxidoreductases
- Discipline
- Analytical, structural and metabolic biochemistry
- Origin
- Inist-CNRS
- Database
- PASCAL
- INIST identifier
- 20272611
Sauf mention contraire ci-dessus, le contenu de cette notice bibliographique peut être utilisé dans le cadre d’une licence CC BY 4.0 Inist-CNRS / Unless otherwise stated above, the content of this bibliographic record may be used under a CC BY 4.0 licence by Inist-CNRS / A menos que se haya señalado antes, el contenido de este registro bibliográfico puede ser utilizado al amparo de una licencia CC BY 4.0 Inist-CNRS
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DOI
10.1016/j.bmc.2008.02.014 
https://dx.doi.org/10.1016/j.bmc.2008.02.014
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